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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC29A1 (1R,13R,14S,15R)-7-(6-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol NA 245470.89 NA NA NA NA BindingDB
SLC29A1 (2R,3R,4S,5R)-2-[6-[(4-tert-butylphenyl)sulfanylmethyl]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol NA 331131.12 NA NA NA NA BindingDB|TTD
SLC29A1 1-[2-[2-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-6-yl]sulfanylphenyl]ethanone NA 446683.59 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3S,4R,5R)-2-(hydroxymethyl)-5-[6-[(2-methylnaphthalen-1-yl)methylsulfanyl]purin-9-yl]oxolane-3,4-diol NA 114815.36 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-[2-amino-6-[(6-methylpyridin-2-yl)methylsulfanyl]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol NA 11481536.21 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-(2-amino-6-propan-2-ylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol NA 190546.07 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-(2-amino-6-ethylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol NA 162181.01 NA NA NA NA BindingDB|TTD
SLC29A1 (2R,3R,4S,5R)-2-[6-[2-[2-[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]ethoxy]ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol NA 912010.84 NA NA NA NA BindingDB|TTD
SLC29A1 Cefepime NA NA NA NA NA 300000 PubChem
SLC29A1 Ceftazidime NA NA NA NA NA 300000 PubChem
SLC29A1 Aztreonam NA NA NA NA NA 400000 PubChem
SLC29A1 Phlorizin 1000000 NA NA NA NA NA PubChem|TTD
SLC29A1 Carumonam NA NA NA NA NA 500000 PubChem
SLC29A1 Doripenem NA NA NA NA NA 300000 PubChem
SLC29A1 Methylthioinosine NA 229086.77 NA NA NA NA BindingDB|TTD
SLC29A1 5-Iodotubercidin NA 229086.77 NA NA NA NA BindingDB|TTD
SLC29A2 Tecadenoson NA|189000 190000|NA NA NA NA NA PubChem
SLC29A2 Uridine 242000|NA NA|234000 NA NA NA NA PubChem
SLC29A2 Adenosine 106000|NA NA|106000 NA NA NA NA PubChem
SLC29A4 Cimetidine 500000 NA NA NA NA NA GtoPDB