GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC29A1 |
(1R,13R,14S,15R)-7-(6-nitro-3,4-dihydro-1H-isoquinolin-2-yl)-11,16-dioxa-2,4,6,9-tetrazatetracyclo[11.2.1.02,10.03,8]hexadeca-3(8),4,6,9-tetraene-14,15-diol |
NA |
245470.89 |
NA |
NA |
NA |
NA |
BindingDB |
SLC29A1 |
(2R,3R,4S,5R)-2-[6-[(4-tert-butylphenyl)sulfanylmethyl]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
331131.12 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
1-[2-[2-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-6-yl]sulfanylphenyl]ethanone |
NA |
446683.59 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-[6-[(2-methylnaphthalen-1-yl)methylsulfanyl]purin-9-yl]oxolane-3,4-diol |
NA |
114815.36 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-[2-amino-6-[(6-methylpyridin-2-yl)methylsulfanyl]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
11481536.21 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-(2-amino-6-propan-2-ylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
190546.07 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-(2-amino-6-ethylsulfanylpurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
162181.01 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
(2R,3R,4S,5R)-2-[6-[2-[2-[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]ethoxy]ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
912010.84 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
SLC29A1 |
Phlorizin |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC29A1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
SLC29A1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC29A1 |
Methylthioinosine |
NA |
229086.77 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A1 |
5-Iodotubercidin |
NA |
229086.77 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC29A2 |
Tecadenoson |
NA|189000 |
190000|NA |
NA |
NA |
NA |
NA |
PubChem |
SLC29A2 |
Uridine |
242000|NA |
NA|234000 |
NA |
NA |
NA |
NA |
PubChem |
SLC29A2 |
Adenosine |
106000|NA |
NA|106000 |
NA |
NA |
NA |
NA |
PubChem |
SLC29A4 |
Cimetidine |
500000 |
NA |
NA |
NA |
NA |
NA |
GtoPDB |