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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC33A1
(5S)-5-[(N-benzoyl)amino]-4-oxo-6-phenyl-hexanoyl-L-tryptophan
195700
NA
NA
NA
NA
NA
TTD
SLC33A1
4-oxidanylidene-4-[[(2~{S})-1-oxidanyl-1-oxidanylidene-propan-2-yl]amino]butanoic acid
NA
1348962.88
NA
NA
NA
NA
TTD
SLC33A1
(2S)-5-(diaminomethylideneamino)-2-(dithiolane-4-carbonylamino)pentanoic acid
NA
113000
NA
NA
NA
NA
TTD
SLC33A1
[(3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl] dithiolane-4-carboxylate
NA
347000
NA
NA
NA
NA
TTD
SLC33A1
Glycylglutamine
NA
7079457.84
NA
NA
NA
NA
TTD
SLC33A1
Retrothiorphan
NA
1000000000
NA
NA
NA
NA
TTD
SLC33A1
(3-Amino-2-oxo-azocan-1-yl)-acetic acid
NA
440000
NA
NA
NA
NA
TTD
SLC33A1
3-Aminohexahydro-2-oxo-1H-azepine-1-acetic acid
NA
480000
NA
NA
NA
NA
TTD
SLC33A1
(2S)-2-[[(2S)-2-[[(3S)-3-amino-2-hydroxydecanoyl]amino]propanoyl]amino]-3-methylbutanoic acid
NA
460000
NA
NA
NA
NA
TTD
SLC33A1
Succinylglycine
NA
1995262.31
NA
NA
NA
NA
TTD
SLC33A1
Phe-Arg
NA
912010.84
NA
NA
NA
NA
TTD
SLC33A1
Arginylphenylalanine
NA
229086.77
NA
NA
NA
NA
TTD
SLC33A1
Aspartylglycine
NA
14125375.45
NA
NA
NA
NA
TTD
SLC33A1
Glycylmethionine
NA
1412537.54
NA
NA
NA
NA
TTD
SLC33A1
Glycyl-L-alanine
NA
1995262.31
NA
NA
NA
NA
TTD
SLC33A1
(3-Amino-2-oxo-piperidin-1-yl)-acetic acid
NA
1700000
NA
NA
NA
NA
TTD
SLC33A1
Histidylleucine
NA
3235936.57
NA
NA
NA
NA
TTD
SLC33A1
1-(4-Carboxy-pentanoyl)-pyrrolidine-2-carboxylic acid
NA
260000
NA
NA
NA
NA
TTD
SLC33A1
(2S)-3-(1H-imidazol-5-yl)-2-(3-sulfanylpropanoylamino)propanoic acid
NA
229086.77
NA
NA
NA
NA
TTD
SLC33A1
Glycylvaline
NA
4570881.9
NA
NA
NA
NA
TTD
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