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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACHE Phenyl-N-(4-aminopiperidine)phosphate NA 5490000 NA NA NA NA BindingDB|TTD
ACHE Triethyl-[2-[2-[[6-oxo-6-[2-(1,2,3,4-tetrahydroacridin-9-yl)hydrazinyl]hexyl]carbamoyl]-4,5-bis[2-(triethylazaniumyl)ethoxy]phenoxy]ethyl]azanium;tribromide;hydrochloride NA 1480000 NA NA NA NA TTD
ACHE Homopiperazine-1,4-bis(methylenephosphonic acid) (11) NA 28720000 NA NA NA NA BindingDB
ACHE 2-[[2-(Isoquinolin-2-ium-2-ylmethyl)phenyl]methyl]isoquinolin-2-ium;dibromide NA 250000 NA NA NA NA TTD
ACHE 1,10-Bis(isoquinolinium)-1,2-phenyldimethylenyl dibromide NA 250000 NA NA NA NA BindingDB
ACHE 1,5-Bis(isoquinolinium)-3-oxapent-1,5-diyl dibromide NA 1310000 NA NA NA NA BindingDB
ACHE (3-Hydroxy-2-methylphenyl)-trimethylazanium NA 141253.75 NA NA NA NA BindingDB|TTD
ACHE Quercetin NA 353860 NA NA NA NA BindingDB|PubChem
ACHE Apigenin 121600 NA NA NA NA NA BindingDB|PubChem
ACHE Scopoletin NA 168600 NA NA NA NA BindingDB|TTD
ACHE Rutin NA|300000 113300|NA NA NA NA NA BindingDB|PubChem
ACHE Umbelliferone NA 29000000 NA NA NA NA BindingDB|TTD
ACHE Fisetin 100200 NA NA NA NA NA BindingDB|PubChem
ACHE 4'-Hydroxychalcone NA 500000 NA NA NA NA TTD
ACHE Rosmarinate NA 1220000 NA NA NA NA BindingDB
ACHE (1S,14S,15S,16S)-5,14-dimethoxy-9-azatetracyclo[7.6.1.02,7.012,16]hexadeca-2,4,6,12-tetraene-4,15-diol NA 200000 NA NA NA NA TTD
ACHE Demethylsuberosin NA 2400000 NA NA NA NA BindingDB|TTD
ACHE 5,7-Dihydroxy-6-methoxy-2-(4-methoxyphenyl)-4-benzopyrone NA 250000 NA NA NA NA TTD
ACHE Peucedanone NA 180000 NA NA NA NA BindingDB|TTD
ACHE 2-(3-Isoquinolin-2-ium-2-ylpropyl)isoquinolin-2-ium;dibromide NA 446000 NA NA NA NA TTD