GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ACHE |
Phenyl-N-(4-aminopiperidine)phosphate |
NA |
5490000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Triethyl-[2-[2-[[6-oxo-6-[2-(1,2,3,4-tetrahydroacridin-9-yl)hydrazinyl]hexyl]carbamoyl]-4,5-bis[2-(triethylazaniumyl)ethoxy]phenoxy]ethyl]azanium;tribromide;hydrochloride |
NA |
1480000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Homopiperazine-1,4-bis(methylenephosphonic acid) (11) |
NA |
28720000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
2-[[2-(Isoquinolin-2-ium-2-ylmethyl)phenyl]methyl]isoquinolin-2-ium;dibromide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
1,10-Bis(isoquinolinium)-1,2-phenyldimethylenyl dibromide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
1,5-Bis(isoquinolinium)-3-oxapent-1,5-diyl dibromide |
NA |
1310000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
(3-Hydroxy-2-methylphenyl)-trimethylazanium |
NA |
141253.75 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Quercetin |
NA |
353860 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ACHE |
Apigenin |
121600 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ACHE |
Scopoletin |
NA |
168600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Rutin |
NA|300000 |
113300|NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ACHE |
Umbelliferone |
NA |
29000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
Fisetin |
100200 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ACHE |
4'-Hydroxychalcone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Rosmarinate |
NA |
1220000 |
NA |
NA |
NA |
NA |
BindingDB |
ACHE |
(1S,14S,15S,16S)-5,14-dimethoxy-9-azatetracyclo[7.6.1.02,7.012,16]hexadeca-2,4,6,12-tetraene-4,15-diol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Demethylsuberosin |
NA |
2400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
5,7-Dihydroxy-6-methoxy-2-(4-methoxyphenyl)-4-benzopyrone |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
ACHE |
Peucedanone |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ACHE |
2-(3-Isoquinolin-2-ium-2-ylpropyl)isoquinolin-2-ium;dibromide |
NA |
446000 |
NA |
NA |
NA |
NA |
TTD |