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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACHE 1-(Quinolin-1-ium-1-ylmethoxymethyl)quinolin-1-ium;dichloride NA 418000 NA NA NA NA TTD
ACHE 1,1''-Prop-2-oxa-1,3-diyl-bis(quinolinium)dichloride NA 418000 NA NA NA NA BindingDB
ACHE [(3R)-3-[methyl(prop-2-ynyl)amino]-2,3-dihydro-1H-inden-5-yl] N-ethyl-N-methylcarbamate;hydrochloride NA 1200000 NA NA NA NA TTD
ACHE NA NA 173000 NA NA NA BindingDB
ACHE NA NA 151300 NA NA NA BindingDB
ACHE NA NA 174000 NA NA NA BindingDB
ACHE Cefepime NA NA NA NA NA 300000 PubChem
ACHE Ceftazidime NA NA NA NA NA 300000 PubChem
ACHE NA NA|640000|2169000 250000|500000|550000|NA NA NA NA BindingDB
ACHE NA NA 107000 NA NA NA BindingDB
ACHE NA NA 150900 NA NA NA BindingDB
ACHE NA NA 111500 NA NA NA BindingDB
ACHE m-Trimethylammonium aniline NA 191866.87 NA NA NA NA TTD
ACHE 1,1-Bis(4-hydroxyiminomethylpyridinium)-methane dibromide NA 2010000 NA NA NA NA BindingDB
ACHE 1-(((4-Carbamoylpyridinium-1-yl)methoxy)methyl)-2-((hydroxyimino)methyl)pyridinium chloride NA NA|203000|460000 200000|800000|NA NA NA NA BindingDB
ACHE N-[3-[(2-chloro-6,7-dimethoxyquinazolin-4-yl)amino]propyl]-5-(dithiolan-3-yl)pentanamide NA 192000 NA NA NA NA BindingDB|TTD
ACHE Bonannione A 120500 NA NA NA NA NA BindingDB
ACHE N-[methoxy-(4-methylphenoxy)phosphoryl]-N-methylmethanamine NA 1730000 NA NA NA NA BindingDB
ACHE N-[dimethylamino-(4-methylphenoxy)phosphoryl]-N-ethylethanamine NA 4930000 NA NA NA NA BindingDB
ACHE [Dimethylamino-(4-methylphenoxy)phosphoryl]formonitrile NA 7530000 NA NA NA NA BindingDB