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drugs and pathways
negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
ACHE
LasR-IN-4
NA
117000
NA
NA
NA
NA
BindingDB
ACHE
Caffeic Acid
NA
5551000
NA
NA
NA
NA
BindingDB
ACHE
Troloxcholine trifluoroacetate (5)
NA
1193000
NA
NA
NA
NA
BindingDB
ACHE
N-propan-2-ylphenothiazine-10-carboxamide
691000
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
N-ethyl-10H-phenothiazine-10-carboxamide
1450000
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
6-Geranyl-4',5,7-trihydroxy-3',5'-dimethoxyflavanone
NA
316300
NA
NA
NA
NA
BindingDB|TTD
ACHE
[2-[3-[7-[Benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-(3-methylphenyl)methanone
NA
102000
NA
NA
NA
NA
BindingDB|TTD
ACHE
5-[4-(1-benzofuran-2-yl)phenoxy]-N-benzyl-N-methylpentan-1-amine
NA
215000
NA
NA
NA
NA
BindingDB|TTD
ACHE
[2-[4-[7-[Benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-naphthalen-1-ylmethanone
NA
101000
NA
NA
NA
NA
BindingDB|TTD
ACHE
NA
NA
106000|210000
NA
NA
NA
BindingDB
ACHE
ethyl (2S,6R)-4-(4-chloroanilino)-1-(4-chlorophenyl)-2,6-diphenyl-3,6-dihydro-2H-pyridine-5-carboxylate
NA
4600000
NA
NA
NA
NA
BindingDB
ACHE
(2E)-N-[(1-benzylpiperidin-4-yl)methyl]-2-hydroxyiminoacetamide
3178000
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
(2E)-N-(1-benzylpiperidin-4-yl)-2-hydroxyiminoacetamide
2430000
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
(NE)-N-[[6-[(1-benzylpiperidin-4-yl)methoxy]pyridin-3-yl]methylidene]hydroxylamine
266000
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
(NE)-N-[[2-[(1-benzylpiperidin-4-yl)methoxy]pyrimidin-5-yl]methylidene]hydroxylamine
198500
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
233800
NA
NA
NA
NA
NA
BindingDB
ACHE
(2E)-N-(1-benzylpiperidin-4-yl)-2-cyano-2-hydroxyiminoacetamide
732500
NA
NA
NA
NA
NA
BindingDB|TTD
ACHE
2303000
NA
NA
NA
NA
NA
BindingDB
ACHE
(2E)-N-[(1-benzylpiperidin-4-yl)methyl]-2-cyano-2-hydroxyiminoacetamide
94963000
NA
NA
NA
NA|NA
NA|NA
BindingDB|TTD
ACHE
NA
566000
NA
NA
NA
NA
BindingDB
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