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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACHE N-methyl-N-[(4-methylphenoxy)-morpholin-4-ylphosphoryl]methanamine NA 13550000 NA NA NA NA BindingDB
ACHE Carbacylamidophosphate, 1b NA 932000 239000 NA NA NA BindingDB
ACHE Carbacylamidophosphate, 4b NA 2890000 4260000 NA NA NA BindingDB
ACHE Aztreonam NA NA NA NA NA 400000 PubChem
ACHE N,N,N-trimethyl-3-nitroanilinium chloride NA 628058.36 NA NA NA NA TTD
ACHE Lysergide NA NA NA NA 104300 NA PubChem
ACHE Sclerone, (+/-)- NA 1080000 NA NA NA NA BindingDB
ACHE [3-(dimethylcarbamoyloxy)-5-[(1R)-1-hydroxy-2-(propan-2-ylamino)ethyl]phenyl] N,N-dimethylcarbamate 390000|710000 NA NA NA NA NA BindingDB
ACHE [2-(dimethylcarbamoyloxy)-4-[(1R)-1-hydroxy-2-(propan-2-ylamino)ethyl]phenyl] N,N-dimethylcarbamate 1200000|1400000 NA NA NA NA NA BindingDB
ACHE Lipoic acid NA 1000000 NA NA NA NA PubChem
ACHE Isonitrosoacetone NA NA 127700 NA NA NA BindingDB
ACHE Diacetylmonoxime NA NA 392600 NA NA NA BindingDB|PubChem
ACHE 4-Morpholineethanamine, N-(4,6-diphenyl-3-pyridazinyl)- NA 260000 NA NA NA NA BindingDB|TTD
ACHE Xanthyletin NA 150000 NA NA NA NA BindingDB|TTD
ACHE (4-Hydroxy-3-methoxyphenyl)(4-morpholinyl)acetonitrile NA 409200 NA NA NA NA BindingDB|TTD
ACHE NA NA|636000|667800|1360000 234000|NA NA NA NA BindingDB
ACHE Carumonam NA NA NA NA NA 500000 PubChem
ACHE 2-(3-Hydroxy-4-methoxyphenyl)-2-(4-methylpiperazin-1-yl)acetonitrile NA 350100 NA NA NA NA BindingDB|TTD
ACHE 2-(4-Hydroxy-3-methoxyphenyl)-2-(4-methylpiperazin-1-yl)acetonitrile NA 340200 NA NA NA NA BindingDB|TTD
ACHE N-Pentyliminobis(methylenephosphonic acid) (4) NA 11660000 NA NA NA NA BindingDB