Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
ACHE | N-methyl-N-[(4-methylphenoxy)-morpholin-4-ylphosphoryl]methanamine | NA | 13550000 | NA | NA | NA | NA | BindingDB |
ACHE | Carbacylamidophosphate, 1b | NA | 932000 | 239000 | NA | NA | NA | BindingDB |
ACHE | Carbacylamidophosphate, 4b | NA | 2890000 | 4260000 | NA | NA | NA | BindingDB |
ACHE | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
ACHE | N,N,N-trimethyl-3-nitroanilinium chloride | NA | 628058.36 | NA | NA | NA | NA | TTD |
ACHE | Lysergide | NA | NA | NA | NA | 104300 | NA | PubChem |
ACHE | Sclerone, (+/-)- | NA | 1080000 | NA | NA | NA | NA | BindingDB |
ACHE | [3-(dimethylcarbamoyloxy)-5-[(1R)-1-hydroxy-2-(propan-2-ylamino)ethyl]phenyl] N,N-dimethylcarbamate | 390000|710000 | NA | NA | NA | NA | NA | BindingDB |
ACHE | [2-(dimethylcarbamoyloxy)-4-[(1R)-1-hydroxy-2-(propan-2-ylamino)ethyl]phenyl] N,N-dimethylcarbamate | 1200000|1400000 | NA | NA | NA | NA | NA | BindingDB |
ACHE | Lipoic acid | NA | 1000000 | NA | NA | NA | NA | PubChem |
ACHE | Isonitrosoacetone | NA | NA | 127700 | NA | NA | NA | BindingDB |
ACHE | Diacetylmonoxime | NA | NA | 392600 | NA | NA | NA | BindingDB|PubChem |
ACHE | 4-Morpholineethanamine, N-(4,6-diphenyl-3-pyridazinyl)- | NA | 260000 | NA | NA | NA | NA | BindingDB|TTD |
ACHE | Xanthyletin | NA | 150000 | NA | NA | NA | NA | BindingDB|TTD |
ACHE | (4-Hydroxy-3-methoxyphenyl)(4-morpholinyl)acetonitrile | NA | 409200 | NA | NA | NA | NA | BindingDB|TTD |
ACHE | NA | NA|636000|667800|1360000 | 234000|NA | NA | NA | NA | BindingDB | |
ACHE | Carumonam | NA | NA | NA | NA | NA | 500000 | PubChem |
ACHE | 2-(3-Hydroxy-4-methoxyphenyl)-2-(4-methylpiperazin-1-yl)acetonitrile | NA | 350100 | NA | NA | NA | NA | BindingDB|TTD |
ACHE | 2-(4-Hydroxy-3-methoxyphenyl)-2-(4-methylpiperazin-1-yl)acetonitrile | NA | 340200 | NA | NA | NA | NA | BindingDB|TTD |
ACHE | N-Pentyliminobis(methylenephosphonic acid) (4) | NA | 11660000 | NA | NA | NA | NA | BindingDB |