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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLCO2A1 Pyruvic Acid 26000000 NA NA NA NA NA BindingDB|PubChem
SLCO2A1 D-Glyceraldehyde 3-Phosphate 15000000 NA NA NA NA NA BindingDB
SLCO2A1 Beta-D-Glucose 6-phosphate 31000000 NA NA NA NA NA BindingDB
SLCO2A1 alpha-D-fructofuranose 1,6-bisphosphate 51000000 NA NA NA NA NA BindingDB|PubChem
SLCO2A1 D-Lactic Acid 48000000 NA NA NA NA NA BindingDB|PubChem
SLCO2A1 Glyceric acid 1,3-biphosphate 57000000 NA NA NA NA NA BindingDB
SLCO2B1 (E)-combretastatin iso A-4 NA 200000 NA NA NA NA TTD
SLCO2B1 Doxorubicin NA|230000 240000|NA NA NA NA NA BindingDB|PubChem|TTD
SLCO2B1 Indomethacin NA|130000 140000|NA NA NA NA NA BindingDB|PubChem|TTD
SLCO2B1 Rutin NA 136900|138038 NA NA NA NA PubChem
SLCO2B1 Pravastatin NA|180000 190000|NA NA NA NA NA BindingDB|PubChem|TTD
SLK 3-[(3-Chloro-4-methoxyphenyl)methylamino]-4-[2-(trifluoromethyl)phenyl]pyrrole-2,5-dione 180000 NA NA NA NA NA BindingDB
SLK 3-[(3-Chloro-4-methoxyphenyl)methylamino]-4-(2-chlorophenyl)pyrrole-2,5-dione 160000 NA NA NA NA NA BindingDB
SMAD2 Gossypol NA NA NA NA 106822 NA PubChem
SMAD2 Miristalkonium chloride NA NA NA NA 19952600|5623410 NA PubChem
SMAD3 1-Cyclohexyl-3-(1-phenylethyl)pyrrolidine-2,5-dione NA 125000 NA NA NA NA BindingDB
SMAD3 Gossypol NA NA NA NA 106822 NA PubChem
SMAD3 Miristalkonium chloride NA NA NA NA 19952600|5623410 NA PubChem
SMARCA4 6-Chloro-3-((4-methylpiperazin-1-yl)methylene)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-one NA NA 417000 NA NA NA BindingDB
SMARCA4 2-(2-chloro-6-fluorophenyl)-2,3-dihydro-1H-quinazolin-4-one NA NA 142000 NA NA NA BindingDB|ChEMBL