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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC7A5 1-Methylhistidine NA 190000 NA NA NA NA PubChem|TTD
SLC7A5 Alloisoleucine, D- NA 3000000 NA NA NA NA TTD
SLC7A5 (2S)-2-amino-3-(1-methyl-1H-1,2,3-triazol-4-yl)propanoic acid NA 1000000 NA NA NA NA TTD
SLC9A1 2-Butyl-2H-benzo[d][1,2,3]triazole NA 101120 NA NA NA NA BindingDB|TTD
SLC9A1 2-(3-Chloropropyl)benzotriazole NA 115250 NA NA NA NA BindingDB|TTD
SLC9A1 2-Heptylbenzotriazole NA 156540 NA NA NA NA BindingDB|TTD
SLC9A1 2-Hexyl-2H-1,2,3-benzotriazole NA 154670 NA NA NA NA BindingDB|TTD
SLC9A1 2-Propylbenzotriazole NA 135000 NA NA NA NA BindingDB|TTD
SLC9A1 2-Pentylbenzotriazole NA 191230 NA NA NA NA BindingDB|TTD
SLC9A1 2-Ethylbenzotriazole NA 355000 NA NA NA NA BindingDB|TTD
SLC9A1 1H-Benzotriazole NA 192680 NA NA NA NA BindingDB|TTD
SLC9A1 2-Methyl-1,2,3-benzotriazole NA 177000 NA NA NA NA BindingDB|TTD
SLC9A2 N-(5-Methyl-1-quinolin-5-yl-1H-pyrazole-4-carbonyl)-guanidine NA 416000 NA NA NA NA BindingDB
SLCO1B1 Verapamil NA 600000 NA NA NA NA PubChem
SLCO1B1 Doxorubicin 150000|NA NA|160000 NA NA NA NA PubChem|TTD
SLCO1B1 Gemfibrozil NA 130000 NA NA NA NA PubChem
SLCO1B3 (E)-combretastatin iso A-4 NA 200000 NA NA NA NA TTD
SLCO1B3 Combretastatin A4 NA 194540 NA NA NA NA TTD
SLCO1B3 Clesacostat NA 137000 NA NA NA NA PubChem
SLCO2A1 Phosphoenolpyruvate 13000000 NA NA NA NA NA BindingDB|PubChem