Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
SLC7A5 | 1-Methylhistidine | NA | 190000 | NA | NA | NA | NA | PubChem|TTD |
SLC7A5 | Alloisoleucine, D- | NA | 3000000 | NA | NA | NA | NA | TTD |
SLC7A5 | (2S)-2-amino-3-(1-methyl-1H-1,2,3-triazol-4-yl)propanoic acid | NA | 1000000 | NA | NA | NA | NA | TTD |
SLC9A1 | 2-Butyl-2H-benzo[d][1,2,3]triazole | NA | 101120 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-(3-Chloropropyl)benzotriazole | NA | 115250 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Heptylbenzotriazole | NA | 156540 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Hexyl-2H-1,2,3-benzotriazole | NA | 154670 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Propylbenzotriazole | NA | 135000 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Pentylbenzotriazole | NA | 191230 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Ethylbenzotriazole | NA | 355000 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 1H-Benzotriazole | NA | 192680 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A1 | 2-Methyl-1,2,3-benzotriazole | NA | 177000 | NA | NA | NA | NA | BindingDB|TTD |
SLC9A2 | N-(5-Methyl-1-quinolin-5-yl-1H-pyrazole-4-carbonyl)-guanidine | NA | 416000 | NA | NA | NA | NA | BindingDB |
SLCO1B1 | Verapamil | NA | 600000 | NA | NA | NA | NA | PubChem |
SLCO1B1 | Doxorubicin | 150000|NA | NA|160000 | NA | NA | NA | NA | PubChem|TTD |
SLCO1B1 | Gemfibrozil | NA | 130000 | NA | NA | NA | NA | PubChem |
SLCO1B3 | (E)-combretastatin iso A-4 | NA | 200000 | NA | NA | NA | NA | TTD |
SLCO1B3 | Combretastatin A4 | NA | 194540 | NA | NA | NA | NA | TTD |
SLCO1B3 | Clesacostat | NA | 137000 | NA | NA | NA | NA | PubChem |
SLCO2A1 | Phosphoenolpyruvate | 13000000 | NA | NA | NA | NA | NA | BindingDB|PubChem |