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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC7A11
(R)-4-Carboxyphenylglycine
NA
1000000
NA
NA
NA
NA
TTD
SLC7A11
5-(Phenylazo)salicylic acid
NA
200000
NA
NA
NA
NA
TTD
SLC7A11
4-[1-[(2,4-Dinitrophenyl)diazenyl]ethyl]-5-methyl-1,2-oxazole-3-carboxylic acid
NA|147000
290000|NA
NA
NA
NA
NA
BindingDB
SLC7A11
5-Methyl-4-[1-[(4-nitrophenyl)diazenyl]ethyl]-1,2-oxazole-3-carboxylic acid
NA
127000
NA
NA
NA
NA
BindingDB
SLC7A11
4-[1-[[3,5-Bis(trifluoromethyl)phenyl]diazenyl]ethyl]-5-methyl-1,2-oxazole-3-carboxylic acid
NA
129000
NA
NA
NA
NA
BindingDB
SLC7A11
4-[1-[(2,4-Dinitrophenyl)diazenyl]ethyl]-5-(2-naphthalen-2-ylethyl)-1,2-oxazole-3-carboxylic acid
NA|113000
225000|NA
NA
NA
NA
NA
BindingDB
SLC7A3
Lysine
NA
158000|NA
NA
NA|158000
NA
NA
PubChem
SLC7A3
Arginine
NA
283000|NA
NA
NA|283000
NA
NA
PubChem
SLC7A5
2-Aminobicyclo[2.2.1]heptane-2-carboxylic acid
NA
112000
NA
NA
NA
NA
TTD
SLC7A5
(2S)-2-Amino-3-(1H-1,2,3-benzotriazol-1-YL)propanoic acid
NA
340000
NA
NA
NA
NA
TTD
SLC7A5
(2R)-2-amino-2-benzyl-4-methylsulfanylbutanoic acid
NA
240000
NA
NA
NA
NA
TTD
SLC7A5
3-[(2S)-2-amino-2-carboxyethyl]-5-methylbenzoic acid
NA
680000
NA
NA
NA
NA
TTD
SLC7A5
(R)-2-Amino-3-(3-(methoxycarbonyl)phenyl)propanoic acid
NA
150000
NA
NA
NA
NA
TTD
SLC7A5
(2S)-2-amino-3-(4-phenyltriazol-1-yl)propanoic acid
NA
1000000
NA
NA
NA
NA
TTD
SLC7A5
(2S)-2-amino-3-[4-(hydroxymethyl)triazol-1-yl]propanoic acid
NA
1000000
NA
NA
NA
NA
TTD
SLC7A5
(2S)-2-amino-3-(4-methyltriazol-1-yl)propanoic acid
NA
440000
NA
NA
NA
NA
TTD
SLC7A5
Poly(1-benzylhistidine)
NA
170000
NA
NA
NA
NA
TTD
SLC7A5
(S)-3-(2-Amino-2-carboxyethyl)benzoic acid
NA
130000
NA
NA
NA
NA
TTD
SLC7A5
L-Alpha-methylphenylalanine
NA
130000
NA
NA
NA
NA
TTD
SLC7A5
3-(2-Pyridyl)-L-alanine
NA
160000
NA
NA
NA
NA
TTD
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