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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACR ethyl 3-[4-(2-phenylbutanoylamino)phenyl]-1H-pyrazole-5-carboxylate NA 3300000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-4-ethylbenzamide NA 210000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-4-methoxybenzamide NA 2210000 NA NA NA NA BindingDB|TTD
ACR 4-(chloromethyl)-N-[4-(diaminomethylideneamino)sulfonylphenyl]benzamide NA 3840000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]butanamide NA 9580000 NA NA NA NA BindingDB|TTD
ACR Ethyl 1-[2-[4-(diaminomethylideneamino)sulfonylanilino]-2-oxoethyl]piperidine-4-carboxylate NA 2990000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-4-fluorobenzamide NA 7110000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-3-(trifluoromethyl)benzamide NA 7050000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-2-(2-methylpiperidin-1-yl)acetamide NA 9900000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-2-(4-methylpiperidin-1-yl)acetamide NA 4980000 NA NA NA NA BindingDB|TTD
ACR 3,4-dichloro-N-[4-(diaminomethylideneamino)sulfonylphenyl]benzamide NA 3800000 NA NA NA NA BindingDB|TTD
ACR 2-bromo-N-[4-(diaminomethylideneamino)sulfonylphenyl]benzamide NA 7630000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-4-ethoxybenzamide NA 130000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]pentanamide NA 1580000 NA NA NA NA BindingDB|TTD
ACR Methyl 1-[2-[4-(diaminomethylideneamino)sulfonylanilino]-2-oxoethyl]piperidine-4-carboxylate NA 9300000 NA NA NA NA BindingDB|TTD
ACR Propyl 1-[2-[4-(diaminomethylideneamino)sulfonylanilino]-2-oxoethyl]piperidine-4-carboxylate NA 3310000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-2-(4-methylphenoxy)acetamide NA 8980000 NA NA NA NA BindingDB|TTD
ACR 2-(4-chlorophenoxy)-N-[4-(diaminomethylideneamino)sulfonylphenyl]acetamide NA 9350000 NA NA NA NA BindingDB|TTD
ACR 2,6-dichloro-N-[4-(diaminomethylideneamino)sulfonylphenyl]benzamide NA 5960000 NA NA NA NA BindingDB|TTD
ACR 3-Methylbutyl 1-[2-[4-(diaminomethylideneamino)sulfonylanilino]-2-oxoethyl]piperidine-4-carboxylate NA 2510000 NA NA NA NA BindingDB|TTD