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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACLY (S)-2-[(R)-6-(5-Chloro-indol-1-yl)-2-hydroxy-hexyl]-2-hydroxy-succinic acid 160000 NA NA NA NA NA BindingDB|TTD
ACLY Ndi-091143 7000000 NA NA NA NA NA BindingDB
ACLY Hydroxycitric acid 300000 NA NA NA NA NA BindingDB
ACP1 Cefsulodin NA 200000 NA NA NA NA PubChem
ACP3 Benzhydrylphosphonic Acid NA 142000 NA NA NA NA BindingDB
ACP3 (Phenyl-p-tolyl-methyl)-phosphonic acid NA 152000 NA NA NA NA BindingDB
ACP3 [(4-Chloro-phenyl)-phenyl-methyl]-phosphonic acid NA 143000 NA NA NA NA BindingDB
ACPP Benzhydrylphosphonic Acid NA 142000 NA NA NA NA TTD
ACPP 9h-Fluoren-9-ylphosphonic acid NA 500000 NA NA NA NA TTD
ACPP (Phenyl-p-tolyl-methyl)-phosphonic acid NA 152000 NA NA NA NA TTD
ACPP [(4-Chloro-phenyl)-phenyl-methyl]-phosphonic acid NA 143000 NA NA NA NA TTD
ACPP Benzylphosphonic Acid NA 500000 NA NA NA NA TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-2-phenoxyacetamide NA 2300000 NA NA NA NA BindingDB|TTD
ACR 5-(2,4-Dichlorophenyl)isoxazole-3-carbaldehyde NA 390000|1700000|39000000 NA NA NA NA BindingDB|TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-3,5-dinitrobenzamide NA 2500000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-3-phenyl-1H-pyrazole-5-carboxamide NA 2800000 NA NA NA NA BindingDB|TTD
ACR N-(3-hydroxypropyl)-3-phenyl-1H-pyrazole-5-carboxamide NA 540000 NA NA NA NA BindingDB|TTD
ACR N-(1-hydroxypropan-2-yl)-3-phenyl-1H-pyrazole-5-carboxamide NA 3000000 NA NA NA NA BindingDB|TTD
ACR Tosyllysine Chloromethyl Ketone NA 142600000 NA NA NA NA TTD
ACR N-[4-(diaminomethylideneamino)sulfonylphenyl]-4-methylbenzamide NA 2060000 NA NA NA NA BindingDB|TTD