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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
USP5 deamino-Cys(1)-D-Phe(4-Et)-Ile-Gln-Asn-Cys(1)-Pro-Leu-Gly-NH2 NA NA 150000 NA NA NA BindingDB
USP5 2-[3-[[2-[5-Cycloheptyl-1-(3,3-dimethyl-2-oxobutyl)-2,4-dioxo-1,3,5-benzotriazepin-3-yl]acetyl]amino]phenyl]acetic acid NA NA 210000 NA NA NA BindingDB
USP5 3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one NA 200000 NA NA NA NA TTD
USP5 3-[5-(2-Bromo-5-methoxyphenyl)-1,3,4-oxadiazol-2-yl]propanoic acid NA NA 270000 NA NA NA BindingDB
USP5 3-[5-(2-Iodophenyl)-1,3,4-oxadiazol-2-yl]propanoic acid NA NA 280000 NA NA NA BindingDB
USP5 3-[5-(2-Bromo-5-fluorophenyl)-1,3,4-oxadiazol-2-yl]propanoic acid NA NA 430000 NA NA NA BindingDB
USP5 1-[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]-2-(pyrrolidin-1-yl)ethan-1-one NA 143400 NA NA NA NA BindingDB
USP5 5-Phenyl-1,3,4-oxadiazole-2-propionic acid NA NA 370000 NA NA NA BindingDB
USP5 3-Benzoylpropionic acid NA NA 680000 NA NA NA BindingDB
USP5 2-(4-Oxo-3,4-dihydroquinazolin-3-yl)acetic acid NA NA 220000 NA NA NA BindingDB
USP5 2-Methyl-4-oxo-4-phenylbutanoic acid NA NA 700000 NA NA NA BindingDB
USP5 3-(2-Thenoyl)propionic acid NA NA 840000 NA NA NA BindingDB
USP5 3-(5-phenyl-2H-tetraazol-2-yl)propanoic acid NA NA 530000 NA NA NA BindingDB
USP5 2-(8-Methyl-4-oxo-3,4-dihydroquinazolin-3-yl)acetic acid NA NA 490000 NA NA NA BindingDB
USP5 (6,7-dimethoxy-4-oxoquinazolin-3(4H)-yl)acetic acid NA NA 110000 NA NA NA BindingDB
USP5 2-(Benzo[d]oxazol-2-yl)acetic acid NA NA 770000 NA NA NA BindingDB
USP5 1-dihydroterritrem B NA NA 150000 NA NA NA BindingDB
USP7 N-[3-[6-amino-4-ethyl-5-(1H-indazol-6-yl)pyridin-3-yl]phenyl]acetamide NA 136000 NA NA NA NA BindingDB
USP7 4-[2-Amino-4-ethyl-5-(3-piperazin-1-ylphenyl)-3-pyridyl]phenol NA 165000 NA NA NA NA BindingDB
USP7 N-[3-[2-amino-4-ethyl-5-(4-hydroxyphenyl)pyridin-3-yl]phenyl]methanesulfonamide NA 118000 NA NA NA NA BindingDB