GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
USP5 |
deamino-Cys(1)-D-Phe(4-Et)-Ile-Gln-Asn-Cys(1)-Pro-Leu-Gly-NH2 |
NA |
NA |
150000 |
NA |
NA |
NA |
BindingDB |
USP5 |
2-[3-[[2-[5-Cycloheptyl-1-(3,3-dimethyl-2-oxobutyl)-2,4-dioxo-1,3,5-benzotriazepin-3-yl]acetyl]amino]phenyl]acetic acid |
NA |
NA |
210000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
USP5 |
3-[5-(2-Bromo-5-methoxyphenyl)-1,3,4-oxadiazol-2-yl]propanoic acid |
NA |
NA |
270000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-[5-(2-Iodophenyl)-1,3,4-oxadiazol-2-yl]propanoic acid |
NA |
NA |
280000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-[5-(2-Bromo-5-fluorophenyl)-1,3,4-oxadiazol-2-yl]propanoic acid |
NA |
NA |
430000 |
NA |
NA |
NA |
BindingDB |
USP5 |
1-[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]-2-(pyrrolidin-1-yl)ethan-1-one |
NA |
143400 |
NA |
NA |
NA |
NA |
BindingDB |
USP5 |
5-Phenyl-1,3,4-oxadiazole-2-propionic acid |
NA |
NA |
370000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-Benzoylpropionic acid |
NA |
NA |
680000 |
NA |
NA |
NA |
BindingDB |
USP5 |
2-(4-Oxo-3,4-dihydroquinazolin-3-yl)acetic acid |
NA |
NA |
220000 |
NA |
NA |
NA |
BindingDB |
USP5 |
2-Methyl-4-oxo-4-phenylbutanoic acid |
NA |
NA |
700000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-(2-Thenoyl)propionic acid |
NA |
NA |
840000 |
NA |
NA |
NA |
BindingDB |
USP5 |
3-(5-phenyl-2H-tetraazol-2-yl)propanoic acid |
NA |
NA |
530000 |
NA |
NA |
NA |
BindingDB |
USP5 |
2-(8-Methyl-4-oxo-3,4-dihydroquinazolin-3-yl)acetic acid |
NA |
NA |
490000 |
NA |
NA |
NA |
BindingDB |
USP5 |
(6,7-dimethoxy-4-oxoquinazolin-3(4H)-yl)acetic acid |
NA |
NA |
110000 |
NA |
NA |
NA |
BindingDB |
USP5 |
2-(Benzo[d]oxazol-2-yl)acetic acid |
NA |
NA |
770000 |
NA |
NA |
NA |
BindingDB |
USP5 |
1-dihydroterritrem B |
NA |
NA |
150000 |
NA |
NA |
NA |
BindingDB |
USP7 |
N-[3-[6-amino-4-ethyl-5-(1H-indazol-6-yl)pyridin-3-yl]phenyl]acetamide |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
USP7 |
4-[2-Amino-4-ethyl-5-(3-piperazin-1-ylphenyl)-3-pyridyl]phenol |
NA |
165000 |
NA |
NA |
NA |
NA |
BindingDB |
USP7 |
N-[3-[2-amino-4-ethyl-5-(4-hydroxyphenyl)pyridin-3-yl]phenyl]methanesulfonamide |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |