Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ADCY5 [2-(6-Amino-purin-9-yl)-ethyl]-hydroxycarbamoylmethyl-carbamic acid tert-butyl ester NA 200000 NA NA NA NA TTD
ADCY5 7-(6-Amino-purin-9-yl)-heptanoic acid ethyl ester NA 200000 NA NA NA NA TTD
ADCY5 2-{[(1R,3R)-3-(6-amino-9H-purin-9-yl)cyclopentyl]oxy}acetic acid NA 200000 NA NA NA NA TTD
ADCY5 2-{[(1R,4R)-4-(6-amino-9H-purin-9-yl)cyclopent-2-en-1-yl]oxy}acetic acid NA 200000 NA NA NA NA TTD
ADCY5 2-{[(1S,3S)-3-(6-amino-9H-purin-9-yl)cyclopentyl]oxy}acetic acid NA 200000 NA NA NA NA TTD
ADCY5 2-[(R)-3-((R)-6-Amino-purin-9-yl)-cyclopentyloxy]-N-hydroxy-acetamide NA 110000 NA NA NA NA BindingDB|TTD
ADCY5 [(R)-3-((R)-6-Amino-purin-9-yl)-cyclopentyloxy]-acetic acid NA 200000 NA NA NA NA TTD
ADCY5 2-{[(1R,4S)-4-(6-amino-9H-purin-9-yl)cyclopent-2-en-1-yl]oxy}-N-hydroxyacetamide NA 102000 NA NA NA NA BindingDB|TTD
ADCY9 (10R,13S,16S,19S)-N-[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-19-(2-amino-2-oxoethyl)-13-benzyl-10-[(4-ethoxyphenyl)methyl]-8,11,14,17,20-pentaoxo-16-propan-2-yl-9,12,15,18,21-pentazaspiro[5.19]pentacosane-22-carboxamide 4400000 NA NA NA NA NA BindingDB
ADH1B N-cyclohexyl-N-methylformamide 920000 NA NA NA NA NA BindingDB
ADH1B N,N-Dicyclopentyl-formamide 1600000 NA NA NA NA NA BindingDB
ADH1B N-cyclopropyl-N-heptyl-formamide 1900000 NA NA NA NA NA BindingDB
ADH1B N,N-Dicyclobutyl-formamide 4900000 NA NA NA NA NA BindingDB
ADH1B N-cyclohexyl-N-propyl-formamide 4000000 NA NA NA NA NA BindingDB
ADH1B N-cyclohexyl-N-cyclopropyl-formamide 250000 NA NA NA NA NA BindingDB
ADH1B N-cyclopentyl-N-cyclopropyl-formamide 4600000 NA NA NA NA NA BindingDB
ADH1B Formamide, N-cyclopentyl-N-propyl-(9CI) 2800000 NA NA NA NA NA BindingDB
ADH1B N-Cyclohexyl-N-ethylformamide 1500000 NA NA NA NA NA BindingDB
ADH1B N-Cyclopentyl-N-Cyclobutylformamide 10000000 NA NA NA NA NA BindingDB
ADH1C N,N-Dicyclopentyl-formamide 1000000 NA NA NA NA NA BindingDB