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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ADRB1 (S)-(+)-5-(1-hydroxy-2-phenethylaminoethyl)-1,3-benzenediol 52178000 NA NA NA NA NA BindingDB
ADRB1 (R)-(-)-5-(1-hydroxy-2-phenethylaminoethyl)-1,3-benzenediol 42466000 NA NA NA NA NA BindingDB
ADRB1 Disodium (R,R)-5-[2-[[2-(3-chlorophenyl)-2-hydroxyethyl]-amino]propyl]-1,3-benzodioxole-2,2-dicarboxylate NA NA NA 111000 NA NA BindingDB
ADRB1 Cefazolin NA NA NA NA NA 300000 PubChem
ADRB1 Meropenem NA NA NA NA NA 300000 PubChem
ADRB1 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-methyl-phosphinic acid 140000 NA NA NA NA NA BindingDB|TTD
ADRB1 (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid monoisopropyl ester 139000 NA NA NA NA NA BindingDB|TTD
ADRB1 2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-malonic acid 243000 NA NA NA NA NA BindingDB|TTD
ADRB1 N-[4-[2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethyl]phenyl]-2-pyridin-2-ylacetamide NA NA NA 120000 NA NA BindingDB|TTD
ADRB1 Terbutaline NA NA 151356 NA NA NA BindingDB
ADRB1 Cefepime NA NA NA NA NA 300000 PubChem
ADRB1 Ceftazidime NA NA NA NA NA 300000 PubChem
ADRB1 Aztreonam NA NA NA NA NA 400000 PubChem
ADRB1 Sematilide NA 7000000 NA NA NA NA BindingDB|TTD
ADRB1 Carumonam NA NA NA NA NA 500000 PubChem
ADRB1 N-[(E)-2-(3-methyl-1,3-benzothiazol-3-ium-2-yl)ethenyl]aniline NA NA 257040 NA NA NA BindingDB
ADRB1 Doripenem NA NA NA NA NA 300000 PubChem
ADRB1 2-(Hydroxymethyl)-4-[1-hydroxy-2-[2-[4-[4-(3-phenylpropyl)piperidin-1-yl]phenyl]ethylamino]ethyl]phenol 125893|125892.54 NA NA NA NA NA BindingDB|TTD
ADRB1 [1-[4-[2-[[2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]ethyl]phenyl]piperidin-4-yl]-phenylmethanone 125893|125892.54 NA NA NA NA NA BindingDB|TTD
ADRB1 N-[4-[1-hydroxy-2-(3-methylimidazol-3-ium-1-yl)ethyl]phenyl]methanesulfonamide;chloride NA 2350000 NA NA NA NA BindingDB|TTD