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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ADRB2 6-Fluoronorepinehprine 1160000 NA NA NA NA NA BindingDB
ADRB2 Imipenem NA NA NA NA NA 300000 PubChem
ADRB2 1-(2-piperidin-1-ylethoxy)-6H-benzo[b][1]benzothiepin-5-one 794328|794328.23 NA NA NA NA NA BindingDB|TTD
ADRB2 2-(1-Hydroxypentyl)-6-methyl-3-(2-phenylethyl)-1H-Indole-5-carboxylic acid NA 1540000 NA NA NA NA BindingDB|TTD
ADRB2 N-(1-benzothiophen-2-ylmethyl)-3-methyloxetan-3-amine 1000000 NA NA NA NA NA TTD
ADRB2 1-(2-methylphenyl)-N-[(4-pyrimidin-2-ylphenyl)methyl]ethanamine 268000 NA NA NA NA NA BindingDB|ChEMBL
ADRB2 4,4,4-trifluoro-N-[[4-(1,3-thiazol-2-yl)phenyl]methyl]butan-2-amine 393000 NA NA NA NA NA BindingDB|ChEMBL
ADRB2 5-[(1S,4S)-1-hydroxy-5-(4-hydroxyphenyl)-4-methylpentyl]benzene-1,3-diol 345000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4R)-1-hydroxy-5-(4-hydroxyphenyl)-4-methylpentyl]benzene-1,3-diol 3695000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4S)-1-hydroxy-5-(4-hydroxyphenyl)-4-methylpentyl]benzene-1,3-diol 10330000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4R)-1-hydroxy-5-(4-hydroxyphenyl)-4-methylpentyl]benzene-1,3-diol 27749000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4S)-1-hydroxy-5-(4-methoxyphenyl)-4-methylpentyl]benzene-1,3-diol 474000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4R)-1-hydroxy-5-(4-methoxyphenyl)-4-methylpentyl]benzene-1,3-diol 1930000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4S)-1-hydroxy-5-(4-methoxyphenyl)-4-methylpentyl]benzene-1,3-diol 5269000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4R)-1-hydroxy-5-(4-methoxyphenyl)-4-methylpentyl]benzene-1,3-diol 15881000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4S)-5-(4-aminophenyl)-1-hydroxy-4-methylpentyl]benzene-1,3-diol 2934000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4R)-5-(4-aminophenyl)-1-hydroxy-4-methylpentyl]benzene-1,3-diol 7937000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4S)-5-(4-aminophenyl)-1-hydroxy-4-methylpentyl]benzene-1,3-diol 23125000 NA NA NA NA NA BindingDB
ADRB2 5-[(1R,4R)-5-(4-aminophenyl)-1-hydroxy-4-methylpentyl]benzene-1,3-diol 28624000 NA NA NA NA NA BindingDB
ADRB2 5-[(1S,4S)-1-hydroxy-4-methyl-5-phenylpentyl]benzene-1,3-diol 1864000 NA NA NA NA NA BindingDB