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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ADRB2 Ceftazidime NA NA NA NA NA 300000 PubChem
ADRB2 4-[1-Hydroxy-2-[[3-[[2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]-2,2-dimethylpropyl]amino]ethyl]-2-(hydroxymethyl)phenol NA 251189|251188.64 NA NA NA NA BindingDB|TTD
ADRB2 Aztreonam NA NA NA NA NA 400000 PubChem
ADRB2 Carumonam NA NA NA NA NA 500000 PubChem
ADRB2 (S,R)-(+)-fenoterol 10330000 NA NA NA NA NA BindingDB
ADRB2 (R,S)-(-)-fenoterol 3695000 NA NA NA NA NA BindingDB
ADRB2 R,R-Fenoterol 345000 NA NA NA NA NA BindingDB
ADRB2 (S,S)-(+)-fenoterol 27749000 NA NA NA NA NA BindingDB
ADRB2 1-(Benzo[b]thiophen-2-yl)-N-methylmethanamine 373000 NA NA NA NA NA BindingDB|ChEMBL
ADRB2 1-(4-Pyridyl)piperazine NA NA 141600 NA NA NA ChEMBL
ADRB2 Doripenem NA NA NA NA NA 300000 PubChem
ADRB2 2-(Hydroxymethyl)-4-[1-hydroxy-2-[2-[4-[4-(3-phenylpropyl)piperidin-1-yl]phenyl]ethylamino]ethyl]phenol 199526 NA NA NA NA NA BindingDB
ADRB2 3-(hydroxymethyl)-5-methyl-2-pentyl-1-phenethyl-1H-indole-6-carboxylic acid NA 280000 NA NA NA NA BindingDB|TTD
ADRB3 4-(3-Hexyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide NA NA NA 56234133 NA NA BindingDB
ADRB3 4-(3-Hexyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide NA NA NA 70794578 NA NA BindingDB
ADRB3 1-ethyl-3-((S)-3-((R)-2-hydroxy-3-(3-(methylsulfonyl)phenoxy) propylamino)-1-oxa-8-azaspiro[4.5]decan-8-ylsulfonyl)quinolin-4(1H)-one NA 107300 NA NA NA NA BindingDB
ADRB3 3-(2-{(R)-2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-thiazol-5-yl)-propionic acid 146000 NA NA NA NA NA BindingDB
ADRB3 N-{4-[2-(2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-4-(3-octyl-2-oxo-imidazolidin-1-yl)-benzenesulfonamide NA NA NA 457088190 NA NA BindingDB
ADRB3 Fenofibrate NA 123945 NA NA NA NA PubChem
ADRB3 (R)-N-(3-(2-amino-1-hydroxyethyl)-2-fluoro-6-hydroxyphenyl)methanesulfonamide 120000 NA NA NA NA NA BindingDB|TTD