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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALAD 2-[2-(Thiophene-2-carbonylamino)ethyl]-3-[[3-(trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD 2-[2-(Thiophene-2-carbonylamino)ethyl]-1-[[3-(trifluoromethyl)phenyl]methyl]benzimidazole-4-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD 2-[2-(Thiophene-2-carbonylamino)ethyl]-3-[[3-(trifluoromethyl)phenyl]methyl]benzimidazole-4-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD 2-[2-(Thiophene-2-carbonylamino)ethyl]-1-[[4-(trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acid NA 637000 NA NA NA NA BindingDB|TTD
ALB 3-(2-bromo-2-chloro-1,1-difluoroethyl)-3H-diazirine NA 800000 NA NA NA NA BindingDB|TTD
ALB 1-Azido-2-bromo-2-chloro-1,1-difluoro-ethane NA 300000 NA NA NA NA BindingDB|TTD
ALB 3-(2-Chloro-1,1,2-trifluoroethyl)-3-fluorodiazirine NA 2200000 NA NA NA NA BindingDB|TTD
ALB 3-Bromo-3-(2-chloro-1,1,2-trifluoroethyl)diazirine NA 700000 NA NA NA NA BindingDB|TTD
ALB Ladarixin 831000 NA NA NA NA NA BindingDB
ALB Biphenyl-3-carboxylic acid 251000 NA NA NA NA NA BindingDB
ALB [4-[2-(Fluoromethoxy)phenyl]phenyl]-imino-methyl-oxo-lambda6-sulfane NA NA 156000 NA NA NA BindingDB
ALB Sulindac 26302700000000 NA NA NA NA NA PubChem
ALB (R)-N-Benzyl-2-(2,5-dioxopyrrolidin-1-yl)propanamide NA NA 1970000 NA NA NA BindingDB
ALB methyl (2S)-2-acetamido-6-[4-(4-iodophenyl)butanoylamino]hexanoate NA NA 110000 NA NA NA BindingDB
ALB 8-[2-(4-Isopropyl-thiazol-2-yl)-ethyl]-3-(1H-tetrazol-5-yl)-pyrido[1,2-a]pyrimidin-4-one NA NA 327000 NA NA NA BindingDB
ALB Vismodegib NA NA 120000|130000 NA NA NA BindingDB|PubChem
ALB Verapamil NA NA 645654 NA NA NA PubChem
ALB Chlorpropamide 39810700000000 NA NA NA NA NA PubChem
ALB Desipramine NA NA 851138 NA NA NA BindingDB|PubChem
ALB Diclofenac 331000 NA NA NA NA NA BindingDB