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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
AKT2 4-Phenylpyrazole NA 135000 NA NA NA NA ChEMBL|TTD
AKT2 1-(8-methyl-7H-purin-6-yl)piperidin-4-amine NA 110000 NA NA NA NA TTD
AKT2 5-Amino-3-methyl-4-phenylpyrazole NA 660000 NA NA NA NA ChEMBL|TTD
AKT3 6-{[(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]formamido}hexanamide NA 1000000 NA NA NA NA TTD
AKT3 N-[6-[[(2R)-6-amino-1-[[6-[[(2R)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]benzamide NA 360000 NA NA NA NA BindingDB|TTD
AKT3 4-[[6-[[(2R)-6-amino-1-[[6-[[(2R)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]carbamoylamino]benzamide NA 900000 NA NA NA NA BindingDB|TTD
ALAD 5-Amino-4-oxohexanoic acid 200000000 NA NA NA NA|NA NA|NA BindingDB|TTD
ALAD 1-[(3-Methylphenyl)methyl]benzimidazole-5-carboxylic acid NA 222000 NA NA NA NA BindingDB|TTD
ALAD 1-[(3-Methoxyphenyl)methyl]benzimidazole-5-carboxylic acid NA 156000 NA NA NA NA BindingDB|TTD
ALAD 1-benzyl-1H-1,3-benzodiazole-5-carboxylic acid NA 213000 NA NA NA NA BindingDB|TTD
ALAD 2-[3-(trifluoromethyl)benzoyl]-3,4-dihydro-1H-benzo[b][1,6]naphthyridine-10-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD wALADin1 NA 739000|740000 NA NA NA NA BindingDB|TTD
ALAD 1H-1,3-benzodiazole-5-carboxylic acid NA 511000 NA NA NA NA BindingDB|TTD
ALAD 1-Methyl-1H-benzimidazole-5-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD 1-[(4-Fluorophenyl)methyl]-2-oxo-3-(pyrimidin-2-ylmethyl)benzimidazole-5-carboxylic acid NA 119000 NA NA NA NA BindingDB|TTD
ALAD 1-[(4-Fluorophenyl)methyl]-2-oxo-3-(2-pyrrolidin-1-ylethyl)benzimidazole-5-carboxylic acid NA 1000000 NA NA NA NA TTD
ALAD 1-[[2-(Trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acid NA 145000 NA NA NA NA BindingDB|TTD
ALAD 1-[[4-(Trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acid NA 173000 NA NA NA NA BindingDB|TTD
ALAD 2-[2-(thiophene-2-carbonylamino)ethyl]-3H-benzimidazole-5-carboxylic acid NA 500000 NA NA NA NA BindingDB|TTD
ALAD 1-[[3-(Trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acid NA 197000 NA NA NA NA BindingDB|TTD