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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALOX15 Halenaquinol Sulfate Sodium NA 200000 NA NA NA NA TTD
ALOX15 {2,6-Di-tert-butyl-4-[1-(3,5-di-tert-butyl-4-carboxymethoxyphenylsulfanyl)-1-methylethylsulfanyl]phenoxy}-acetic acid NA 125000 NA NA NA NA TTD
ALOX15 15-Oxo-puupehenoic Acid NA 150000 NA NA NA NA TTD
ALOX15 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine NA 213000 NA NA NA NA BindingDB|TTD
ALOX15 2-(4-chloro-2-methylphenoxy)-N-(2-hydroxy-5-isopropylphenyl)acetamide NA 200000 NA NA NA NA TTD
ALOX5 4-[(2-hydroxy-3-methoxyphenyl)methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide NA 200000 NA NA NA NA TTD
ALOX5 4-Methylquinoline-8-thiol NA 200000 NA NA NA NA TTD
ALOX5 5-Methylquinoline-8-thiol NA 200000 NA NA NA NA TTD
ALOX5 6-Methyl-8-mercaptochinolin NA 200000 NA NA NA NA TTD
ALOX5 Atractylenolide II NA 200000 NA NA NA NA TTD
ALOX5 Ethyl 2-(2-fluorophenyl)-5-hydroxybenzofuran-3-carboxylate NA 116900 NA NA NA NA BindingDB
ALOX5 1-(Benzyloxy)hept-2-yn-4-ol NA 760000 NA NA NA NA BindingDB|TTD
ALOX5 2-Pyridin-2-ylmethyl-1,2-dihydro-indazol-3-one NA NA NA 133000 NA NA BindingDB
ALOX5 1-(4-Methoxy-phenyl)-tetrahydro-pyridazin-3-one NA 156000 NA NA NA NA BindingDB|TTD
ALOX5 1-(4-Ethyl-phenyl)-tetrahydro-pyridazin-3-one NA 125000 NA NA NA NA BindingDB|TTD
ALOX5 1-p-Tolyl-tetrahydro-pyridazin-3-one NA 277000 NA NA NA NA BindingDB|TTD
ALOX5 Atractylenolide Iii NA 200000 NA NA NA NA TTD
ALOX5 7-Hydroxy-8-methyl-3-(4-nitrophenyl)-4H-1-benzopyran-4-one NA 300000 NA NA NA NA BindingDB
ALOX5 3-Methyl-8-quinolinethiol NA 200000 NA NA NA NA TTD
ALOX5 2-(1H-Indol-3-ylmethyl)-1,2-dihydro-indazol-3-one NA NA NA 113000 NA NA BindingDB