GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
6-Phosphonohexanoic acid |
7000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
Phenylsulfanylmethyl-phosphonothioic acid |
460000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
6-Thiophosphono-hexanoic acid methyl ester |
330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
Benzyl-phosphonothioic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
3-chloro-N-[[5-[(4-chlorophenyl)methylsulfanyl]-1,3,4-oxadiazol-2-yl]methyl]aniline |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-benzyl-3-chloro-4-(2-ethoxyanilino)-1H-pyrrole-2,5-dione |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-(Anilinocarbonyl)phenyl 1-benzofuran-2-carboxylate |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-(4-Methoxyphenyl)-4-[(2-phenylvinyl)sulfonyl]piperazine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-[(E)-2-(4-hydroxyphenyl)-1-ethenyl]-5-(methoxycarbonyl)-1,3,3-trimethyl-3H-indolium |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
methyl 2-[(E)-2-(2-hydroxyphenyl)ethenyl]-1,3,3-trimethylindol-1-ium-5-carboxylate;iodide |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-[2-(dibenzylamino)ethyl]-5-methoxy-N-methylindole-2-carboxamide;hydrochloride |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-Thiophosphono-hexanoic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
11-Oxo-11 h-pyrido[2,1-b]quinazoline-7-carboxylic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxylic acid |
NA |
710000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2-{[5-[(2,6-dimethylphenoxy)methyl]-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]thio}-N-1,3-thiazol-2-ylacetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-Hydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2,3-Dimethoxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
410000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2,3-Dihydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
N-[(1-benzyl-1H-benzimidazol-2-yl)methyl]-1-[2-(diethylamino)ethyl]-1H-benzimidazol-2-amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-[[1-[2-(1,3-Benzodioxol-5-yloxy)ethyl]indol-3-yl]methylidene]-1,3-diazinane-2,4,6-trione |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |