GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
3-(3-bromo-5-ethoxy-4-hydroxyphenyl)-2-cyano-N-(4-hydroxyphenyl)acrylamide |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2-(2H-tetrazol-5-yl)-12H-benzo[g]pyrido[2,1-b]quinazolin-12-one |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2-methyl-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2,3-dimethoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
6-(2H-tetrazol-5-yl)-13,15-dioxa-2,8-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1(17),2,4,6,10,12(16)-hexaen-9-one |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-(5-Chlorothiophen-2-yl)-2-(6-ethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-(1,3-Benzodioxol-5-yl)-5-[(2,4-dichlorophenyl)methylsulfanyl]tetrazole |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N,N'-dibenzyl-4-chloro-1,3-benzenedisulfonamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
Methylphosphonic acid |
11000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ALPG |
|
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
N-(2-chlorophenyl)-4-methyl-2-[[(E)-3-phenylprop-2-enoyl]amino]-1,3-thiazole-5-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-amino-6-methyl-4-oxo-4H-chromene-3-carbaldehyde |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-(4-Methylphenyl)-3-((3-(trifluoromethyl)benzyl)sulfanyl)-2-thiophenecarboxamide |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
6,7-Diacetoxy-4-methylcoumarin |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
ethyl 2-{3-[(4,6-dioxo-2-thioxotetrahydro-5(2H)-pyrimidinylidene)methyl]-2,5-dimethyl-1H-pyrrol-1-yl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-(3,4-dihydroxyphenyl)-2-{[1-(4-methoxyphenyl)-1H-tetrazol-5-yl]sulfanyl}ethanone |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-(5-Bromofuran-2-yl)-5-[(2-chlorophenoxy)methyl]-1,2,4-oxadiazole |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |