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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPG 3-(3-bromo-5-ethoxy-4-hydroxyphenyl)-2-cyano-N-(4-hydroxyphenyl)acrylamide NA NA NA 999000 NA NA BindingDB
ALPG 3-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 620000 NA NA NA NA BindingDB
ALPG 2-(2H-tetrazol-5-yl)-12H-benzo[g]pyrido[2,1-b]quinazolin-12-one NA 230000 NA NA NA NA BindingDB
ALPG 2-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 140000 NA NA NA NA BindingDB
ALPG 8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 280000 NA NA NA NA BindingDB
ALPG 2-methyl-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 210000 NA NA NA NA BindingDB
ALPG 2,3-dimethoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 340000 NA NA NA NA BindingDB
ALPG 6-(2H-tetrazol-5-yl)-13,15-dioxa-2,8-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1(17),2,4,6,10,12(16)-hexaen-9-one NA 230000 NA NA NA NA BindingDB
ALPG 1-(5-Chlorothiophen-2-yl)-2-(6-ethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-(1,3-Benzodioxol-5-yl)-5-[(2,4-dichlorophenyl)methylsulfanyl]tetrazole NA NA NA 999000 NA NA BindingDB
ALPG N,N'-dibenzyl-4-chloro-1,3-benzenedisulfonamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG Methylphosphonic acid 11000000 NA NA NA NA NA BindingDB|PubChem
ALPG NA 999000 NA NA NA NA BindingDB
ALPG N-(2-chlorophenyl)-4-methyl-2-[[(E)-3-phenylprop-2-enoyl]amino]-1,3-thiazole-5-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 2-amino-6-methyl-4-oxo-4H-chromene-3-carbaldehyde NA NA NA 999000 NA NA BindingDB
ALPG N-(4-Methylphenyl)-3-((3-(trifluoromethyl)benzyl)sulfanyl)-2-thiophenecarboxamide NA 999000 NA NA NA NA BindingDB
ALPG 6,7-Diacetoxy-4-methylcoumarin NA NA NA 999000 NA NA BindingDB
ALPG ethyl 2-{3-[(4,6-dioxo-2-thioxotetrahydro-5(2H)-pyrimidinylidene)methyl]-2,5-dimethyl-1H-pyrrol-1-yl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate NA NA NA 999000 NA NA BindingDB
ALPG 1-(3,4-dihydroxyphenyl)-2-{[1-(4-methoxyphenyl)-1H-tetrazol-5-yl]sulfanyl}ethanone NA NA NA 999000 NA NA BindingDB
ALPG 3-(5-Bromofuran-2-yl)-5-[(2-chlorophenoxy)methyl]-1,2,4-oxadiazole NA NA|999000 NA 999000|NA NA NA BindingDB