Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ABCB1 Dihydroergocristine 511000 NA NA NA NA NA PubChem
ABCB1 1-(2-Hydroxy-3-isopropylamino-propyl)-5-methyl-2-phenyl-4-(thiophene-2-carbonyl)-1,2-dihydro-pyrazol-3-one NA NA NA 123030 NA NA TTD
ABCB1 Dihydroergocryptine 360500 NA NA NA NA NA PubChem
ABCB1 Methyleugenolglycol NA NA NA 500000 NA NA TTD
ABCB1 3-((2-Phenethylphenoxy)methyl)pyridine NA NA NA 125000 NA NA TTD
ABCB1 1-(Benzyloxy)-2-(2-phenylethyl)benzene NA NA NA 1000000 NA NA TTD
ABCB1 3-((2-(3-Methoxyphenethyl)phenoxy)methyl)pyridine NA NA NA 1000000 NA NA TTD
ABCB1 4-iodo-1-methyl-N'-[(1-methyl-1H-pyrazol-5-yl)carbonyl]-1H-pyrazole-3-carbohydrazide NA NA NA 500000 NA NA TTD
ABCB1 Erythromycin 1000000 NA NA NA NA NA PubChem
ABCB1 Vinblastine 140000 NA NA NA NA NA PubChem
ABCB1 (E)-3-(3-bromo-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one NA 500000 NA NA NA NA TTD
ABCB1 (E)-3-(3-iodo-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one NA 500000 NA NA NA NA TTD
ABCB1 N-tert-butyl-N'-[(E)-(2-hydroxy-3-methoxyphenyl)methylideneamino]oxamide NA NA NA 102200 NA NA TTD
ABCB1 2-Ethoxyethyl 4-aminobenzoate NA NA NA 311800 NA NA TTD
ABCB1 N'-benzoyl-N-tert-butyl-3,5-dimethylbenzohydrazide NA 100400 NA NA NA NA TTD
ABCB1 Troleandomycin 483300 NA NA NA NA NA PubChem
ABCB1 Dexpropranolol NA 583000 NA NA NA NA TTD
ABCB1 Verapamil NA 224000|446500|168200|303530 NA NA NA NA PubChem
ABCB1 Celiprolol 313000 NA NA NA NA NA PubChem
ABCB1 1-[2-(2-Hydroxy-3-morpholin-4-ylpropoxy)phenyl]ethanone NA NA NA 207000 NA NA TTD