| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ABCB1 |
5-(2,6-Ditert-butylselenopyran-1-ium-4-yl)thiophene-2-carboxylic acid;hexafluorophosphate |
NA |
111000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB1 |
(E)-4-(3-oxo-3-(3,4,5-trimethoxyphenyl)prop-1-en-1-yl)benzoic acid |
NA |
141253.75 |
NA |
NA |
NA |
NA |
TTD |
| ABCB1 |
Vincristine |
213000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| ABCB1 |
Progesterone |
NA |
192200 |
NA |
NA |
NA |
NA |
PubChem |
| ABCB1 |
Atorvastatin |
NA |
307000|271000 |
NA |
NA |
NA |
NA |
PubChem |
| ABCB1 |
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB1 |
(4Z)-2,5-dimethyl-4-[phenyl(propylamino)methylene]-2,4-dihydro-3H-pyrazol-3-one |
NA |
NA |
NA |
272500 |
NA |
NA |
TTD |
| ABCB1 |
2-Amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d][1,3]thiazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB1 |
Oseltamivir |
NA |
1300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB1 |
2-(1-azepanyl)-N'-(2-chloro-6-fluorobenzylidene)-2-oxoacetohydrazide |
NA |
NA |
NA |
159300 |
NA |
NA |
TTD |
| ABCB1 |
(3S,6S,9S,12R,15S,18R,21R,24R,30S,33S)-12-(4-aminobutyl)-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhept-4-enyl]-1,4,7,10,15,19,25,28-octamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undecone |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB1 |
Levopropranolol |
170000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
N-(1-adamantylmethyl)-2-chloro-5-(piperazin-1-ylmethyl)benzamide |
NA |
124000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
Moxifloxacin Hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
(S)-2-[[6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(1-methylethyl)-2,4-dioxothieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-isoxazolidinol |
NA |
703000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
Emetine |
NA |
135000|133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
6-((3,5-dimethyl-1H-pyrazol-4-yl)methyl)-5-((4S)-4-hydroxy-1,2-oxazolidine-2-carbonyl)-3-methyl-1-(2-methylpropyl)-1H,2H,3H,4H-thieno(2,3-d)pyrimidine-2,4-dione |
NA |
247800 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
Dihydralazine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Hexylcaine Hydrochloride |
NA |
505700 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Propylene Glycol |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |