| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BACE1 |
N-methyl-N-{2-methyl-5-[(6-phenylpyrimidin-4-yl)amino]phenyl}methanesulfonamide |
NA |
1600000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
N-[5-({6-[2-(dimethylamino)phenyl]pyrimidin-4-yl}amino)-2-methylphenyl]methanesulfonamide |
NA |
317000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
N-(2-methyl-5-{[6-(2-methylphenyl)pyrimidin-4-yl]amino}phenyl)methanesulfonamide |
NA |
219000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
(2-Chloro-6-fluorophenyl)methyl carbamimidothioate |
NA |
NA |
300000|350000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
4H-3,1-Benzothiazin-2-amine |
NA |
790000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
3-(2-amino-5-chloro-1H-benzimidazol-1-yl)propan-1-ol |
NA |
770000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Byakangelicol |
NA |
104900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
8-Hydroxybergapten |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
1,4-Diamino-2,3-bis[(4-ethylphenyl)sulfanyl]anthracene-9,10-dione |
NA |
253000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
3-Methyl-2-(2-(2-methyl-5-phenylfuran-3-carboxamido)acetamido)butanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
7-Prenyloxycoumarin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
Coumarin |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| BACE1 |
Oxypeucedanin |
NA |
359200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Marmesin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
8-Bromoquinolin-2-amine |
NA |
NA|562000 |
540000|NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Latifolin |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Hydroxyamfetamine |
NA |
NA |
800000 |
NA |
NA |
NA |
PubChem |
| BACE1 |
3-Methyl-2-[[2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]acetyl]amino]butanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
2,11-Dimethyl-4,9-dioxo-3,5,8,10-tetraazadodecane-1,12-dioic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
N-(6-chloropyridin-3-yl)-4-fluorobenzamide |
NA |
NA |
114000 |
NA |
NA |
NA |
BindingDB|ChEMBL |