| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BACE1 |
2,3,4,5-tetra(3,4,5-trihydroxyphenylcarbonyloxy)-6-(3,4,5-trihydroxyphenylcarbonyloxymethyl)-(2R,3S,4R,5S,6S)-tetrahydro-2H-pyran |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
4-(2-Aminoethyl)-2-phenylphenol |
NA |
NA |
350000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-[(2S,3S)-4-[[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl]amino]-3-hydroxy-1-phenylbutan-2-yl]-3-methylsulfonylbenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
N-[(2S,3R)-4-[[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl]-methylamino]-3-hydroxy-1-phenylbutan-2-yl]-3-methylsulfonylbenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
N-[(2R,3S)-1-[[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl]amino]-2-hydroxy-5-methylhexan-3-yl]-3-methylsulfonylbenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
3-[2-(3-{[(Furan-2-ylmethyl)(methyl)amino]methyl}phenyl)ethyl]pyridin-2-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
N-(1-adamantyl)-2-[3-cyano-4-(4-fluorophenyl)-6-phenylpyridin-2-yl]sulfanylacetamide |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
3-(3-Chlorobenzyl)-5-isobutyl-5-methyl-2-iminohydantoin |
NA |
NA |
123000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
(2Z)-3-(3-chlorobenzyl)-2-imino-5,5-dimethylimidazolidin-4-one |
NA |
NA |
200000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
2-Ethylhex-2-enyl carbamimidothioate |
NA |
NA |
550000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
7-Bromoquinolin-2-amine |
NA |
NA|460000 |
266000|NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
5-(4-Morpholino-3-(p-tolylcarbamoyl)phenylamino)-5-oxopentanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Heraclenin |
NA |
443600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
6,7-Furano-5-prenyloxy hydrocoumaric acid |
NA |
185600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
6,7-Furano-5-prenyloxy hydrocoumaric acid methyl ester |
NA |
203300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
6,7-Furano-8a-methoxy-5-prenyloxy hydrocoumaric acid |
NA |
203300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Xestosaprol F |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Xestosaprol G |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Xestosaprol I |
NA |
163000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
Xestosaprol M |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |