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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(2-morpholinoethyl)pentanamide NA 440000 NA NA NA NA BindingDB|TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(cyclopropylmethyl)pentanamide NA 243000 NA NA NA NA BindingDB|TTD
BACE1 (3S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(2-(pyrrolidin-3-yl)ethyl)pentanamide NA 270000 NA NA NA NA BindingDB|TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(cyclohexylmethyl)-N-methylpentanamide NA 375000 NA NA NA NA BindingDB|TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-((tetrahydro-2H-pyran-4-yl)methyl)pentanamide NA 1000000 NA NA NA NA TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(pyridin-2-ylmethyl)pentanamide NA 1000000 NA NA NA NA TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(3-fluorobenzyl)pentanamide NA 340000 NA NA NA NA BindingDB|TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(4-fluorobenzyl)pentanamide NA 264000 NA NA NA NA BindingDB|TTD
BACE1 (S)-methyl 2-((S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)pentanamido)-3-tert-butoxypropanoate NA 168000 NA NA NA NA BindingDB|TTD
BACE1 5-[3-(3,5-Bis-trifluoromethyl-phenyl)-ureido]-2-dimethylamino-N-(3-methoxy-propyl)-benzamide NA 283900 NA NA NA NA BindingDB
BACE1 Bergaptol NA 500000 NA NA NA NA TTD
BACE1 Esculetin NA 500000 NA NA NA NA TTD
BACE1 Umbelliferone NA 500000 NA NA NA NA TTD
BACE1 N-((2S,3R)-4-(1-(4-tert-butyloxazol-2-yl)cyclohexylamino)-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl)acetamide NA 137800 NA NA NA NA BindingDB|TTD
BACE1 Demethylsuberosin NA 412900 NA NA NA NA BindingDB|TTD
BACE1 Osthenol NA 500000 NA NA NA NA TTD
BACE1 6-(4-Chlorophenyl)quinolin-2-amine NA NA 2000000 NA NA NA BindingDB
BACE1 6-Cyclohexylquinolin-2-amine NA NA 296000 NA NA NA BindingDB
BACE1 7H-Furo(3,2-g)(1)benzopyran-7-one, 4,9-dihydroxy- NA 500000 NA NA NA NA TTD
BACE1 N-[3-[(5S,7S)-3-amino-5-methyl-7-phenyl-6,7-dihydro-2H-1,4-oxazepin-5-yl]-4-fluorophenyl]-5-chloropyridine-2-carboxamide NA 142000 NA NA NA NA BindingDB|TTD