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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BACE1 4-(6-Oxo-7,7-diphenylheptanamido)butanoic acid NA 500000 NA NA NA NA BindingDB|TTD
BACE1 2-(2,4-Dichlorobenzylamino)-2-oxoethyl 2-hydroxy-3-methoxybenzoate NA 500000 NA NA NA NA BindingDB|TTD
BACE1 3-(2-(4-(2-Hydroxyethylamino)-6-morpholino-1,3,5-triazin-2-yl)hydrazinyl)-3-phenylpropanoic acid NA 500000 NA NA NA NA BindingDB|TTD
BACE1 2-(2-((4-ethyl-8-methyl-2-oxo-2H-chromen-7-yloxy)carbonylamino)acetamido)acetic acid NA 500000 NA NA NA NA BindingDB|TTD
BACE1 CID 46927332 NA 200000 NA NA NA NA BindingDB
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-5-methyl-N-(pyridin-2-ylmethyl)hexanamide NA 235000 NA NA NA NA BindingDB|TTD
BACE1 3-(Pyridin-4-yl)imidazo[1,2-a]pyrimidine NA 1008000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-benzylbutanamide NA 1403000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-isopropylbutanamide NA 193000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(2-morpholinoethyl)butanamide NA 827000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(2-(pyrrolidin-3-yl)ethyl)butanamide NA 444000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(pyridin-2-ylmethyl)butanamide NA 426000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(1-methylpiperidin-4-yl)butanamide NA 325000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(3-fluorobenzyl)butanamide NA 249000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(cyclopropylmethyl)butanamide NA 2854000 NA NA NA NA BindingDB|TTD
BACE1 4-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-(3-fluorobenzyl)-N-methylbutanamide NA 194000 NA NA NA NA BindingDB|TTD
BACE1 (R)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-benzylpentanamide NA 516000 NA NA NA NA BindingDB|TTD
BACE1 (R)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-isopropyl-5-methylhexanamide NA 1000000 NA NA NA NA TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-isopropyl-5-methylhexanamide NA 246000 NA NA NA NA BindingDB|TTD
BACE1 (S)-3-(2-amino-5-chloro-1H-benzo[d]imidazol-1-yl)-N-isopropylpentanamide NA 695000 NA NA NA NA BindingDB|TTD