Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| BACE1 | Mormin | NA | 103500 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Demethoxycurcumin | NA | 1600000 | NA | NA | NA | NA | BindingDB |
| BACE1 | Didemethyl Curcumin | NA | 2200000 | NA | NA | NA | NA | BindingDB |
| BACE1 | Morusinol | NA | 135900 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Cyclomorusin | NA | 101200 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Neocyclomorusin | NA | 146100 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | 5-methyl-4H-1,3,4-thiadiazin-2-amine | NA | 8200000 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Tyramine | NA | NA | 2000000 | NA | NA | NA | BindingDB|PubChem |
| BACE1 | (3s)-Spiro[indole-3,3'-Pyrrolidin]-2(1h)-One | NA | NA|1100000 | 1400000|NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Methyl (3s,5'r)-2-Oxo-1,2-Dihydrospiro[indole-3,3'-Pyrrolidine]-5'-Carboxylate | NA | 242000 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | Tetrahydro-2h-Pyran-4-Yl (3s,5'r)-2-Oxo-1,2-Dihydrospiro[indole-3,3'-Pyrrolidine]-5'-Carboxylate | NA | 114000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| BACE1 | [(3R)-3-benzylmorpholin-4-yl]-[(3S,4R)-4-phenylpyrrolidin-3-yl]methanone | NA | 240000 | NA | NA | NA | NA | BindingDB|TTD |
| BACE1 | 4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-9-hydroxyfuro[3,2-g]chromen-7-one | NA | 500000 | NA | NA | NA | NA | TTD |
| BACE1 | 2-amino-3-methyl-6-[(1S,2S)-2-phenylcyclopropyl]pyrimidin-4-one | NA | 2000000 | NA | NA | NA | NA | TTD |
| BACE1 | Lomatin | NA | 500000 | NA | NA | NA | NA | TTD |
| BACE1 | Psoralen | NA | 500000 | NA | NA | NA | NA | PubChem|TTD |
| BACE1 | 4-Hydroxy-dextroamphetamine | NA | NA | 800000 | NA | NA | NA | BindingDB |
| BACE1 | 9-Hydroxy-4-(3,7-dimethyl-2,6-octadienyloxy)-psoralen | 102700 | NA | NA | NA | NA | NA | BindingDB |
| BACE1 | Xanthotoxol | NA | 500000 | NA | NA | NA | NA | TTD |
| BACE1 | Xanthyletin | NA | 500000 | NA | NA | NA | NA | TTD |