| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BACE1 |
N-Substituted tetramic acid, 93 |
NA |
184000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 94 |
NA |
258000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 95 |
NA |
265000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 96 |
NA |
241000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 97 |
NA |
459000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 98 |
NA |
424000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 99 |
NA |
212000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
N-Substituted tetramic acid, 100 |
NA |
139000000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
NH2-Thr-Asn-Ile-Lys-Thr-Glu-Glu-Ile-Ser-Glu-Val-Asn-Leu-Gly-Ala-Glu-Phe-Arg |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
2-Chloro-5-(5-((2-(4-(phenylamino)-6-(piperidin-1-yl)-1,3,5-triazin-2-yl)hydrazono)methyl)furan-2-yl)benzoic acid |
NA |
151800 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
Columbianetin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
Curcumin |
NA |
343000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| BACE1 |
6-Methylquinolin-2-amine |
NA |
NA |
1600000 |
NA |
NA |
NA |
BindingDB |
| BACE1 |
Phellopterin |
NA |
1432000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE2 |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| BACE2 |
3-{2-[(5-Aminopentyl)amino]-2-oxoethoxy}-5-({[1-(4-fluorophenyl)ethyl]amino}carbonyl)phenyl phenylmethanesulfonate |
NA |
137000 |
NA |
NA |
NA |
NA |
TTD |
| BACE2 |
3-(benzylsulfonylamino)-N-[(2S,3R)-4-[[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl]amino]-3-hydroxy-1-phenylbutan-2-yl]benzamide |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| BACE2 |
3-(benzylsulfonyl)-N-((2S,3R)-4-((S)-1-(cyclohexylamino)-1-oxopropan-2-ylamino)-3-hydroxy-1-phenylbutan-2-yl)benzamide |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| BACE2 |
3-(N-benzyl-N-methylsulfamoyl)-N-((2S,3R)-4-((S)-1-(cyclohexylamino)-1-oxopropan-2-ylamino)-3-hydroxy-1-phenylbutan-2-yl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BACE2 |
9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |