| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BAZ2B |
N-(1-acetylindol-3-yl)-N-(5-methoxy-2-methylphenyl)-3-(trifluoromethyl)benzamide |
NA |
NA |
140000 |
NA |
NA |
NA |
BindingDB |
| BAZ2B |
Methylpyrrolidone |
NA |
34000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| BAZ2B |
N,1,5-trimethyl-1H-pyrazole-3-carboxamide |
NA |
1094000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
N-methyl-6-phenylnicotinamide |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
N-methyl-2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carboxamide |
NA |
241000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
N-(5-Oxo-5,6,7,8-tetrahydronaphthalen-2-yl)acetamide |
NA |
476000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
2-methyl-1H-imidazole-4-carbothioamide |
NA |
495000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
Pyrazinethiocarboxamide |
NA |
NA|190000 |
524000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
2-Acetyl-8-fluoro-2,3,4,5-tetrahydro-1H-pyrido[4,3-B]indole |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
8-Chloro-1,3,4,5-tetrahydropyrido[4,3-b]indole-2-carbothioamide |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| BAZ2B |
3-(2-acetyl-8-chloro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)-N-methylpropanamide |
NA |
143000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
1-(8-Amino-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)ethanone |
NA |
NA |
336000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| BAZ2B |
N-(2-acetyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-8-yl)methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| BAZ2B |
1-(8-Nitro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)ethanone |
NA |
NA |
694000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| BAZ2B |
2-(2-acetyl-8-chloro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BAZ2B |
1-[8-(Methylamino)-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl]ethanone |
NA |
NA |
274000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| BAZ2B |
2-methyl-N-(1-thieno[3,2-b]pyridin-6-ylethyl)pyridin-3-amine |
NA |
481000 |
NA |
NA |
NA |
NA |
BindingDB |
| BAZ2B |
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-methylpyridin-3-amine |
NA |
490000 |
NA |
NA |
NA |
NA |
BindingDB |
| BAZ2B |
N-(1,1-dioxothian-3-yl)-2-methylpyridin-3-amine |
NA |
279000 |
NA |
NA |
NA |
NA |
BindingDB |
| BAZ2B |
Ro 22-3581 |
NA |
826000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |