| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCAT2 |
5-methyl-4-oxo-N-pyridin-3-yl-3H-thieno[2,3-d]pyrimidine-6-carboxamide |
NA |
251188.64 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCAT2 |
2-hydroxy-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide |
NA |
1258925.41 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
3,5-dimethyl-6-(piperidine-1-carbonyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one |
NA |
630957.34 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
(2-Hydroxy-2-phenylethyl)urea |
NA |
794328.23 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCAT2 |
3-Phenylthiophene-2-carboxamide |
NA |
158489.32 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCAT2 |
2,1,3-Benzothiadiazol-5-ylmethanol |
NA |
1258925.41 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
2-(1,2-Benzoxazol-3-yl)acetic acid |
NA |
1258925.41 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
1,2,3,4-Tetrahydro-3-methyl-8-quinolinesulfonamide |
NA |
1258925.41 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
N-(Pyrimidin-5-Yl)benzamide |
NA |
1e+06|1000000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCAT2 |
Benzanilide |
NA |
630957.34 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
2-methylsulfonyl-N-phenylbenzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCAT2 |
5-Ethyl-2-Methyl-7-Oxo-4,7-Dihydropyrazolo[1,5-A]pyrimidine-3-Carbonitrile |
NA |
630957.34 |
NA |
NA |
NA |
NA |
TTD |
| BCAT2 |
(1,1'-Biphenyl)-2-carboxamide |
NA |
158489.32 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BCHE |
[2-((5aS,7R,9aS)-1-Formyl-7-hydroxy-4-methoxy-6,7-dihydro-5aH-dibenzofuran-9a-yl)-ethyl]-methyl-carbamic acid ethyl ester |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(6R)-6-[(3S,5R,7S,10S,13R,14R,17R)-3,7-dihydroxy-4,4,10,13,14-pentamethyl-11,15-dioxo-2,3,5,6,7,12,16,17-octahydro-1H-cyclopenta[a]phenanthren-17-yl]-2-methyl-4-oxoheptanoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
1-[(E)-benzylideneamino]-3-pyridin-4-ylurea |
NA|685200 |
845200|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
ethyl (1S,12S,14R)-14-hydroxy-9-methoxy-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6(17),7,9,15-tetraene-4-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
9alpha-Hydroxyandrost-4-ene-3,17-dione |
NA |
141280 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-Methoxylonchocarpin |
NA |
101910 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
3,4,9,10,11,12-Hexahydro-2H-benzothieno[3,2-e]pyrimido[1,2-c]pyrimidine (12) |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |