| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCL2L1 |
2-[3-(2-Methoxyphenyl)acryloyl]-7-(methylamino)-2,4,6-cycloheptatrien-1-one |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
alpha-(3-(Dimethylamino)propyl)-alpha-phenylbenzenemethanol |
NA |
NA |
5000000 |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
4-amino-N-(1,3-benzoxazol-2-yl)benzenesulfonamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2,3,5,6-Tetrakis(furan-2-yl)pyrazine |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-(5-methylfuran-2-yl)-N-(5-methylpyridin-2-yl)quinoline-4-carboxamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-2-(2-thienyl)acetamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-Amino-3-benzyloxypyridine |
NA |
NA |
691800 |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Ethyl 2-Amino-6-(3'',5''-dimethoxyphenyl)-4-(2-ethoxy-2-oxoethyl)-4H-chromene-3-carboxylate |
1236000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-Amino-6-bromo-4-(cyano-ethoxycarbonyl-methyl)-4H-chromene-3-carboxylic acid ethyl ester |
659600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Ethyl 4-(1-cyano-2-ethoxy-2-oxoethyl)-2-imino-3,4-dihydrochromene-3-carboxylate |
570000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Ethyl 4-(2-ethoxy-2-oxoethyl)-2-imino-6-phenyl-3,4-dihydrochromene-3-carboxylate |
343800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
1-(6-chloranyl-1,3-benzothiazol-2-yl)-2-(furan-2-yl)-3-(furan-2-ylcarbonyl)-4-oxidanyl-2H-pyrrol-5-one |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(1R,9S,10S,12S,14E,16S,19R,20R,21S,22R)-9,21-dihydroxy-5,10,12,14,16,20,22-heptamethyl-23,24-dioxatetracyclo[17.3.1.16,9.02,7]tetracosa-5,7,14-triene-3,4-dione |
NA |
NA |
528000|1830000 |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(1R,12S,16S,19R,20R,21S,22R)-4,8,21-Trihydroxy-10-(S)-methyl-5,12,14,16,20,22-hexamethyl-23-oxa-tricyclo[17.3.1.0*2,7*]tricosa-2(7),4,14-triene-3,6,9-trione |
NA |
NA|230000 |
10800000|NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(1R,2S,4S,6E,8S,11R,12R,13S,14R,15R,22R)-13-hydroxy-1'',2,4,6,8,12,14,19-octamethyl-23,25,26,27-tetraoxaspiro[pentacyclo[18.5.1.1^{11,15}.0^{1,22}.0^{16,21}]heptacosane-24,4''-piperidine]-6,16(21),19-triene-17,18-dione |
NA |
NA |
377000|399000 |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(2S)-2-[[(2S)-4-amino-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-5-amino-2-[(2-aminoacetyl)amino]-5-oxopentanoyl]amino]-3-methylbutanoyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-oxopentanoyl]amino]propanoyl]amino]propanoyl]amino]-3-methylpentanoyl]amino]-3-methylpentanoyl]amino]acetyl]amino]-3-carboxypropanoyl]amino]-3-carboxypropanoyl]amino]-3-methylpentanoyl]amino]-4-oxobutanoyl]amino]-5-(diaminomethylideneamino)pentanoic acid |
NA |
NA |
NA |
270000 |
NA |
NA |
BindingDB |
| BCL2L1 |
ethyl 2-amino-6-ethyl-4-(1-cyano-2-ethoxy-2-oxoethyl)-4Hchromene-3-carboxylate |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
ethyl 2-amino-6-methyl-4-(1-cyano-2-ethoxy-2-oxoethyl)-4Hchromene-3-carboxylate |
191000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
[2-oxo-2-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)amino]ethyl] (E)-3-(5-bromofuran-2-yl)prop-2-enoate |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |