| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCL2L1 |
(E)-3-(furan-2-yl)-N,N-dipyridin-2-ylprop-2-enamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-[(6,7-Dihydroxy-2-oxochromen-4-yl)methylsulfanyl]-3-(3-methoxyphenyl)quinazolin-4-one |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
4-(4-Chlorophenyl)-1-[(3s)-3,4-Dihydroxybutyl]-N-[3-(4-Methylpiperazin-1-Yl)propyl]-3-Phenyl-1h-Pyrrole-2-Carboxamide |
NA|138000 |
453000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
4-[[(2R)-4-(dimethylamino)-1-phenylsulfanylbutan-2-yl]amino]-3-nitro-N-phenylbenzenesulfonamide |
NA|166000 |
547000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(3-formylphenyl) (E)-3-(furan-2-yl)prop-2-enoate |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
5-(4-chlorophenyl)-1,2-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-phenylpyrrole-3-carboxamide |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
5-[[2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetyl]amino]-2-hydroxybenzoic acid |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
N-[5-(3,4-Dimethoxy-benzyl)-[1,3,4]thiadiazol-2-yl]-2-thiophen-2-yl-acetamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-[[5-(furan-2-yl)-4-propan-2-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
3,6,7-Trimethyl-benzofuran-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2L1 |
4-[2-[(E)-[2,4-dioxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidin-5-ylidene]methyl]pyrrol-1-yl]benzoic acid |
NA |
103947 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
8-(2-Furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrile |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
6-[(4-Fluorophenyl)methyl]-2-(furan-2-ylmethylidene)-[1,3]thiazolo[3,2-b][1,2,4]triazine-3,7-dione |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |