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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCL2L1 N-[3-methyl-1,1-bis(oxidanylidene)thiolan-3-yl]-3-(4-oxidanylidene-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)propanamide NA 108803 NA NA NA NA BindingDB
BCL2L1 N-[2-(2,3-dimethylanilino)-2-oxoethyl]-3-pyrrol-1-ylbenzamide NA 108803 NA NA NA NA BindingDB
BCL2L1 N-(2-((2,5-Dimethylphenyl)amino)-2-oxoethyl)-N-methyl-3-(1H-pyrrol-1-yl)benzamide NA 108803 NA NA NA NA BindingDB
BCL2L1 N-[1-[3-[(4-chlorobenzoyl)amino]phenyl]ethylideneamino]-2,5-dihydroxybenzamide NA 108803 NA NA NA NA BindingDB
BCL2L1 Chlorcyclizine NA NA 700000 NA NA NA BindingDB|PubChem
BCL2L1 4-(4-Fluorophenyl)benzoic acid NA NA 300000|3e+05 NA NA NA BindingDB|ChEMBL
BCL2L1 2-[5-(3,4-Dimethylphenyl)-4-oxo-3-thieno[2,3-d]pyrimidinyl]acetonitrile NA 108803 NA NA NA NA BindingDB
BCL2L1 3-[(2-nitrophenyl)sulfanylmethyl]-4-prop-2-enyl-1H-1,2,4-triazole-5-thione NA 108803 NA NA NA NA BindingDB
BCL2L1 3-Benzylsulfanyl-5,6-bis(furan-2-yl)-1,2,4-triazine NA 108803 NA NA NA NA BindingDB
BCL2L1 Mcl1-IN-1 NA 108803 NA NA NA NA BindingDB
BCL2L1 as-Triazine, 5,6-di-2-furyl-3-(methylthio)- NA 108803 NA NA NA NA BindingDB
BCL2L1 2-Hydroxy-N-(1,8,8-trimethyl-2,4-dioxo-3-aza-bicyclo[3.2.1]oct-3-yl)-benzamide NA 108803 NA NA NA NA BindingDB
BCL2L1 3,7-Dimethyl-1-benzofuran-2-carboxylic acid 1000000 NA NA NA NA NA TTD
BCL2L1 N-(2,4-difluorophenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamide NA 108803 NA NA NA NA BindingDB
BCL2L1 5-[(5-Bromo-2-methoxyphenyl)methylidene]-2-(furan-2-yl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one NA 108803 NA NA NA NA BindingDB
BCL2L1 N-(4-chloro-2,5-dimethoxyphenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamide NA 108803 NA NA NA NA BindingDB
BCL2L1 methyl 2-[(5,6-dihydro-4H-cyclopenta[d]isoxazol-3-ylcarbonyl)amino]benzoate NA 108803 NA NA NA NA BindingDB
BCL2L1 2-[5-(2,5-Dihydroxyphenyl)sulfonylnaphthalen-1-yl]sulfonylbenzene-1,4-diol NA 108803 NA NA NA NA BindingDB
BCL2L1 Gossypol NA NA 338000 NA NA NA BindingDB|PubChem
BCL2L1 4-(2-Furyl)-6-(4-methylphenyl)-2-oxo-1,2-dihydro-3-pyridinecarbonitrile NA 108803 NA NA NA NA BindingDB