| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCL2L1 |
3-({7-[(2-Furylmethyl)thio]-4-nitro-2,1,3-benzoxadiazol-5-yl}amino)propyl acetate |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
4-[(4-Chlorophenyl)methylsulfamoyl]-1-hydroxynaphthalene-2-carboxylic acid |
338000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
1-Hydroxy-4-(naphthalen-1-ylsulfamoyl)naphthalene-2-carboxylic acid |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-hydroxy-4-(N-isobutylphenyl-sulfonamido) benzoic acid |
154000|154181 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
3-(4-chloro-3-nitrophenyl)-N-[4-(1-pyrrolidinyl)phenyl]acrylamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(2~{R})-2-[[6-ethyl-5-(1~{H}-indol-4-yl)thieno[2,3-d]pyrimidin-4-yl]amino]-3-phenyl-propanoic acid |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
1-(3,4-Dihydroxyphenyl)-2-[(4-prop-2-enyl-5-pyridin-3-yl-1,2,4-triazol-3-yl)sulfanyl]ethanone |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-(4-Bromoanilino)-6-nitro-1,3-benzothiazin-4-one |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Sodium;2-nitro-4-(3-nitro-4-oxidophenyl)sulfonylphenolate |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(2S)-2-[[6-ethyl-5-(4-methylsulfanylphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]propanoic acid |
216000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
(2R)-2-[[5-(3-hydroxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]propanoic acid |
287000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
(2R)-2-[[6-ethyl-5-(3-hydroxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2-phenylacetic acid |
319000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
(2S)-2-[[6-ethyl-5-(3-hydroxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2-phenylacetic acid |
107000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCL2L1 |
|
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(6E)-2-(2-furyl)-5-imino-6-[[1-(4-methoxyphenyl)pyrrol-2-yl]methylene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-[(5E)-5-[[2-[(2-chlorophenyl)methoxy]-5-nitrophenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(E)-3-(4-chloro-3-nitro-phenyl)-2-(5-pyrrolidinosulfonyl-2-thienyl)acrylic acid |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
N-(4-ethoxy-3-morpholinosulfonyl-phenyl)-3-pyrrol-1-yl-benzamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
3,4-Dimethoxybenzoic acid [2-[(5-nitro-2-thiazolyl)amino]-2-oxoethyl] ester |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-[(5Z)-5-[1-[2-(3-bromoanilino)-2-oxoethyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]ethanesulfonic acid |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |