| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCL2 |
ethyl (2S)-2-[(5Z)-5-[[4-[[4-[(Z)-[3-[(2S)-1-ethoxy-1-oxo-3-phenylpropan-2-yl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]phenoxy]methoxy]phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate |
226000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-[(2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoyl]oxyethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate |
243000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-[2-[(2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoyl]oxyethoxy]ethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
4-[[(2R)-4-(dimethylamino)-1-phenylsulfanylbutan-2-yl]amino]-3-nitro-N-(4-piperazin-1-ylphenyl)benzenesulfonamide |
138000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
3,6,7-Trimethyl-benzofuran-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
5,6,7,8-Tetrahydro-1-naphthol |
NA |
4300000 |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
5-[(1-naphthylmethyl)sulfanyl]-1H-1,2,4-triazole |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
Chelerythrine Chloride |
171000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
3-Chloro-6-methyl-1-benzothiophene-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
3,4-Dichloro-1-benzothiophene-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-(4-Chloro-3-methylphenoxy)acetic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2L1 |
[2-(3-Chlorophenyl)-5-(furan-2-yl)pyrazol-3-yl]-piperidin-1-ylmethanone |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
2-[(4,4-Dimethyl-2,6-dioxocyclohexyl)-(5-ethyl-4-nitrothiophen-2-yl)methyl]-5,5-dimethylcyclohexane-1,3-dione |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Terephthalamide scaffold, 47 |
450000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Terephthalamide scaffold, 41 |
138000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
1-Phenyl-1H-pyrazolo[3,4-d]pyrimidine |
NA |
NA |
4000000 |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Terephthalamide scaffold, 43 |
780000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
(R)-4-((4-(Dimethylamino)-1-(phenylthio)butan-2-yl)amino)-3-nitrobenzenesulfonamide |
NA |
238000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
Terephthalamide scaffold, 42 |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2L1 |
N-(2-furanylmethyl)-2-(4-oxo-6-phenyl-3-thieno[2,3-d]pyrimidinyl)acetamide |
NA |
108803 |
NA |
NA |
NA |
NA |
BindingDB |