| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
1-(1-Hexadecyltriazol-4-yl)cyclohexan-1-ol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[1-(3-Chlorophenyl)triazol-4-yl]cyclohexan-1-ol |
NA |
512000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
Methyl 2-[4-[4-(1-hydroxycyclohexyl)triazol-1-yl]phenyl]acetate |
NA |
568000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[1-(3-Nitrophenyl)triazol-4-yl]cyclohexan-1-ol |
NA |
585000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
[4-(1-Hydroxycyclohexyl)triazol-1-yl] benzoate |
NA |
248000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[1-(4-Chlorophenyl)triazol-4-yl]cyclohexan-1-ol |
NA |
294000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[2-(4-Phenyltriazol-1-yl)phenyl]ethanone |
NA |
295000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-(1-(4-Bromophenyl)-1h-1,2,3-triazol-4-yl)cyclohexanol |
NA |
297600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
|
NA |
1620000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(dimethylamino)ethyl N-(2-chloropyridin-4-yl)carbamate;trihydrochloride |
379700 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
2-(dimethylamino)ethyl N-(3-bromopyridin-4-yl)carbamate;dihydrochloride |
273400 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
triethyl-[2-[2-[2-[(1R,4S,5R,9S,10R,13S)-5,9,13-trimethyl-14-oxotetracyclo[11.2.1.01,10.04,9]hexadecane-5-carbonyl]oxyethoxy]ethoxy]ethyl]azanium;bromide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
N'-[(Z)-(4-bromo-2-fluorophenyl)methylidene]-2-hydroxybenzohydrazide (26) |
NA |
451600 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-Carbamoyl-1-(3-(4-((hydroxyimino)methyl)pyridinium-1-yl)propyl)pyridinium bromide |
660000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1-Butyl-5,5-dimethyl-2-(nitrosomethyl)-4,6-dihydropyrimidine |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
N,N-dimethyl-2-nitroso-N'-pentylethanimidamide |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
N'-benzyl-N,N-dimethyl-2-nitrosoethanimidamide |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(6-Aminohexylideneamino)naphthalene-1,4-diol |
NA |
294000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-carbamoyl-1-(4-(4-((E)-(hydroxyimino)methyl)pyridinium-1-yl)but-2-enyl)pyridinium bromide |
910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
5-[1,2]Dithiolan-3-yl-pentanoic acid [3-(4-{3-[ethyl-(2-methoxy-benzyl)-amino]-propylamino}-3,6-dioxo-cyclohexa-1,4-dienylamino)-propyl]-amide |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB |