| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
Galantamine |
NA |
9400000|18600000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| BCHE |
N'-[2-[2-(6-aminohexylamino)ethyldisulfanyl]ethyl]hexane-1,6-diamine |
NA |
645654 |
NA |
NA |
NA |
NA |
BindingDB |
| BCL2 |
Isosclerone |
474760 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-[5-(4-Bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl]propanoic acid |
115000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
(2S)-2-[[6-ethyl-5-(4-methylsulfanylphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]propanoic acid |
359000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
(2R)-2-[[6-ethyl-5-(3-hydroxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2-phenylacetic acid |
470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
(2S)-2-[(6-ethyl-5-phenylthieno[2,3-d]pyrimidin-4-yl)amino]propanoic acid |
418000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
(2S)-2-[[6-ethyl-5-[3-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidin-4-yl]amino]propanoic acid |
437000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
(2S)-2-[[6-ethyl-5-(3-hydroxyphenyl)thieno[2,3-d]pyrimidin-4-yl]amino]-2-phenylacetic acid |
269000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
7-methyl-3-phenyl-1H-indole-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
Propanoic acid, 3-(4-chloro-3,5-dimethylphenoxy)- |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
Antimycin A3 |
124000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| BCL2 |
2-[5-(4-Bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl]-glutaric acid |
320000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
4-(4-Fluorophenyl)benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
3,7-Dimethyl-1-benzofuran-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-Propenyl 2-[5-(4-bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl]-3-propanoate |
192000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-Propenyl 2-[5-(4-bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl]-3-phenylpropanoate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
prop-2-enyl (2S)-2-(5-benzhydrylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl)-3-phenylpropanoate |
260000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
ethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate |
260000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCL2 |
2-[2-[2-[(2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoyl]oxyethoxy]ethoxy]ethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate |
161000 |
NA |
NA |
NA |
NA |
NA |
TTD |