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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCHE 3-[4-(1-benzofuran-2-yl)phenoxy]-N-benzyl-N-methylpropan-1-amine NA 136000 NA NA NA NA BindingDB|TTD
BCHE 1-(3-Nitrophenyl)-4-phenyl-1H-1,2,3-triazole NA 499000 NA NA NA NA BindingDB|TTD
BCHE 1-(4-Bromophenyl)-4-phenyl-1H-1,2,3-triazole NA 375300 NA NA NA NA BindingDB|TTD
BCHE 1-[(E)-(4-methoxyphenyl)methylideneamino]-3-pyridin-4-ylurea NA|624425 786500|NA NA NA NA NA BindingDB|TTD
BCHE 1-[(E)-(3,4-dimethoxyphenyl)methylideneamino]-3-pyridin-4-ylurea NA|282620 426400|NA NA NA NA NA BindingDB|TTD
BCHE NA|446480 528400|NA NA NA NA NA BindingDB
BCHE Pyridostigmine Bromide NA 16000000 NA NA NA NA PubChem
BCHE Benzo[c]thiophen-1(3H)-one 4894000 NA NA NA NA NA BindingDB|TTD
BCHE Edrophonium Chloride NA 1370000 NA NA NA NA PubChem|TTD
BCHE Huperzine A NA 10000000 NA NA NA NA PubChem
BCHE 7-nitro-3H-2-benzothiophen-1-one 341000 NA NA NA NA NA BindingDB|TTD
BCHE Thioctic Acid NA 1000000 NA NA NA NA PubChem
BCHE 1-[1-(2-Nitrophenyl)triazol-4-yl]cyclohexan-1-ol NA 333300 NA NA NA NA BindingDB|TTD
BCHE Methyl 2-[4-(1-hydroxycyclohexyl)triazol-1-yl]acetate NA 362300 NA NA NA NA BindingDB|TTD
BCHE 1-(1-Pyridin-4-yltriazol-4-yl)cyclohexan-1-ol NA 384600 NA NA NA NA BindingDB|TTD
BCHE 1-[1-(4-Nitrophenyl)triazol-4-yl]cyclohexan-1-ol NA 409000 NA NA NA NA BindingDB|TTD
BCHE 1-[1-(2-Chlorophenyl)triazol-4-yl]cyclohexan-1-ol NA 430000 NA NA NA NA BindingDB|TTD
BCHE 1-[3-(4-Phenyl-1H-1,2,3-triazol-1-yl)phenyl]ethanone NA 451000 NA NA NA NA BindingDB|TTD
BCHE 1-[3-[4-(1-Hydroxycyclohexyl)triazol-1-yl]phenyl]ethanone NA 452000 NA NA NA NA BindingDB|TTD
BCHE 1-Hexadecyl-4-phenyltriazole NA 454500 NA NA NA NA BindingDB|TTD