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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCHE 20-Hydroxyecdysone NA 1050000 NA NA NA NA BindingDB
BCHE n-Butyl ganoderate H NA 200000 NA NA NA NA TTD
BCHE N'-[(Z)-(3-bromophenyl)methylidene]-2-hydroxybenzohydrazide (19) NA 121320 NA NA NA NA BindingDB
BCHE 1-(((4-Carbamoylpyridinium-1-yl)methoxy)methyl)-2-((hydroxyimino)methyl)pyridinium chloride 215000 NA NA NA NA NA BindingDB
BCHE 2-Hydroxy-N'-{(Z)-[4-(trifluoromethyl)phenyl]methylidene} benzohydrazide (18) NA 213250 NA NA NA NA BindingDB
BCHE 2-Hydroxy-N'-{(Z)-[3-(trifluoromethyl)phenyl]methylidene} benzohydrazide (14) NA 112230 NA NA NA NA BindingDB
BCHE N-[3-[(2-chloro-6,7-dimethoxyquinazolin-4-yl)amino]propyl]-5-(dithiolan-3-yl)pentanamide NA 205000 NA NA NA NA BindingDB|TTD
BCHE 2-(4-Methylphenyl)-5,6,7,8-tetrahydrofuro[2,3-b]quinolin-4-amine NA 119000 NA NA NA NA BindingDB|TTD
BCHE 1-[(2R,4S,5R)-4-[(6,8-ditert-butyl-5-fluoro-2-oxo-4H-1,3,2lambda5-benzodioxaphosphinin-2-yl)oxy]-5-(hydroxymethyl)oxolan-2-yl]-5-iodopyrimidine-2,4-dione NA 3000000 NA NA NA NA TTD
BCHE N-Butyl Lucidenate N NA 200000 NA NA NA NA TTD
BCHE 7-Methoxy-9-[7-(7-methoxy-1,2,3,4-tetrahydroacridin-9-yl)-1,7-diazacyclododec-1-yl]-1,2,3,4-tetrahydroacridine NA 656000 NA NA NA NA BindingDB|TTD
BCHE N-Butyl Lucidenate A NA 200000 NA NA NA NA TTD
BCHE Ganoderic Acid Y NA 200000 NA NA NA NA TTD
BCHE Methyl Ganoderate A Acetonide NA 200000 NA NA NA NA TTD
BCHE 11alpha-Hydroxytestolactone, 6 NA 283950 NA NA NA NA BindingDB
BCHE Carbacylamidophosphate, 1b NA 9980000 5063000 NA NA NA BindingDB
BCHE Carbacylamidophosphate, 4b NA 16720000 33557000 NA NA NA BindingDB
BCHE Lipoic acid NA 1000000 NA NA NA NA PubChem|TTD
BCHE (2E)-1-(4-aminophenyl)-3-(4-methoxyphenyl)prop-2-en-1-one NA 119000 NA NA NA NA BindingDB|TTD
BCHE NA|212400 245800|NA NA NA NA NA BindingDB