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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCL2L1 2,3-Dihydro-1,4-benzodioxin-3-yl-[4-(4-methoxyphenyl)sulfonylpiperazin-1-yl]methanone NA 108803 NA NA NA NA BindingDB
BCL2L1 (E)-3-amino-2-[2-[[5-(isopropylamino)-1,3,4-thiadiazol-2-yl]thio]acetyl]but-2-enenitrile NA 108803 NA NA NA NA BindingDB
BCL2L1 2-(1-Iminoethyl)-4-[[5-(3-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-3-oxobutanenitrile NA 108803 NA NA NA NA BindingDB
BCL2L1 (4R,12aR)-4,7-bis(dimethylamino)-10,12a-dihydroxy-1,3,11,12-tetraoxo-4,4a,5,5a,6,11a-hexahydrotetracene-2-carboxamide NA 108803 NA NA NA NA BindingDB
BCL2L1 [4,4-Bis-(4-chloro-phenyl)-but-3-enyl]-dimethyl-amine NA 180000 NA NA NA NA BindingDB|TTD
BCL2L1 Resveratrol NA 190000 NA NA NA NA BindingDB|PubChem|TTD
BCL2L1 ent-Trachyloban-18-oic acid NA 400000 NA NA NA NA BindingDB|TTD
BCL2L1 ent-17-Hydroxytrachyloban-18-oic acid NA 220000 NA NA NA NA BindingDB|TTD
BCL2L1 ent-16alpha-Hydroxykaur-11-en-18-oic acid NA 380000 NA NA NA NA BindingDB|TTD
BCL2L1 N-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamide NA 108803 NA NA NA NA BindingDB
BCL2L1 3-(4-Ethoxyphenyl)-8-(furan-2-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile NA 108803 NA NA NA NA BindingDB
BCL2L1 N-[3-(3,4-dihydro-2H-pyrrol-5-ylsulfamoyl)phenyl]-2-(furan-2-yl)quinoline-4-carboxamide NA 108803 NA NA NA NA BindingDB
BCL2L1 Isokaempferide NA 108803 NA NA NA NA BindingDB
BCL2L1 1,1-Bis(4-chlorophenyl)-4-(dimethylamino)butan-1-ol NA NA 450000 NA NA NA BindingDB
BCL2L1 (R)-1-(4-chlorophenyl)-4-(dimethylamino)-1-phenylbutan-1-ol NA NA 500000 NA NA NA BindingDB
BCL2L1 4-phenoxy-N-(4-phenylphenyl)sulfonylbenzamide NA 161300 NA NA NA NA BindingDB|TTD
BCL2L1 3-(3,4-dimethoxyphenyl)-N-(4-phenoxyphenyl)sulfonylbenzamide NA 1000000 NA NA NA NA TTD
BCL2L1 NA 108803 NA NA NA NA BindingDB
BCL2L1 N-(6-Bromo-benzothiazol-2-yl)-2-(3-cyano-7-hydroxy-5-oxo-4,5-dihydro-thieno[3,2-b]pyridin-2-ylsulfanyl)-acetamide NA 108803 NA NA NA NA BindingDB
BCL2L1 methyl 2-{[(6,7-dihydroxy-2-oxo-2H-chromen-4-yl)methyl]amino}benzoate NA 108803 NA NA NA NA BindingDB