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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCL2L2 prop-2-enyl (2S)-2-(5-benzhydrylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl)-3-phenylpropanoate 116000 NA NA NA NA NA BindingDB|TTD
BCL2L2 ethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate 116000 NA NA NA NA NA BindingDB|TTD
BCL2L2 2-[(2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoyl]oxyethyl (2S)-2-[(5Z)-5-[(4-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanoate 101000 NA NA NA NA NA BindingDB|TTD
BCL2L2 BH3I-1 124000 NA NA NA NA NA BindingDB|TTD
BCL2L2 Chelerythrine Chloride 106000 NA NA NA NA NA TTD
BCL2L2 2-Amino-6-bromo-4-(cyano-ethoxycarbonyl-methyl)-4H-chromene-3-carboxylic acid ethyl ester 210000 NA NA NA NA NA BindingDB
BCL2L2 Ethyl 4-(1-cyano-2-ethoxy-2-oxoethyl)-2-imino-3,4-dihydrochromene-3-carboxylate 696610 NA NA NA NA NA BindingDB
BCL2L2 ethyl 2-amino-6-ethyl-4-(1-cyano-2-ethoxy-2-oxoethyl)-4Hchromene-3-carboxylate 120520 NA NA NA NA NA BindingDB
BCL2L2 ethyl 2-amino-6-methyl-4-(1-cyano-2-ethoxy-2-oxoethyl)-4Hchromene-3-carboxylate 198980 NA NA NA NA NA BindingDB
BCL6 Amanozine NA NA 1200000 NA NA NA ChEMBL
BCL6 2-{6-({[2-(1H-indol-3-yl)ethyl]carbamothioyl}amino)-3-[(4-methylpiperazin-1-yl)methyl]-1H-indol-1-yl}-N-(propan-2-yl)acetamide NA 142000 NA NA NA NA TTD
BCL6 2-[(4Z)-4-(5-bromo-2-oxo-1H-indol-3-ylidene)-2-sulfanylidene-1,3-thiazolidin-3-yl]butanedioic acid NA 212000 NA NA NA NA TTD
BCL6 2-[[2-[6-[2-(1H-indol-3-yl)ethylcarbamothioylamino]-3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]acetyl]amino]acetic acid NA 112000 NA NA NA NA TTD
BCL6 2-[[2-[6-[2-(1H-indol-3-yl)ethylcarbamothioylamino]indol-1-yl]acetyl]amino]acetic acid NA 170000 NA NA NA NA TTD
BCL6 2-Chloranyl-4-(cyclopropylmethylamino)pyridine-3-carbonitrile NA 207000 NA NA NA NA TTD
BCL6 N4-phenylpyrimidine-2,4-diamine NA NA 3e+06 NA NA NA ChEMBL
BCL6 N-(2-phenylethyl)-N'-pyridin-3-ylthiourea NA NA 3200000 NA NA NA ChEMBL
BCL6 2-[(5Z)-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanedioic acid NA 212000 NA NA NA NA TTD
BCL6 Rifamycin NA NA 1000000 NA NA NA PubChem
BCL6 4-(Benzylamino)-2-chloronicotinonitrile NA 120000 NA NA NA NA TTD