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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
BCR 4-[4-(5-Bromo-2-morpholin-4-ylpyrimidin-4-yl)piperazin-1-yl]sulfonylbenzonitrile NA 500000 NA NA NA NA TTD
BCR 5-Bromo-2-chloro-4-(4-cyclopropylsulfonylpiperazin-1-yl)pyrimidine NA 500000 NA NA NA NA TTD
BCR [4-(5-Bromo-2-morpholin-4-ylpyrimidin-4-yl)piperazin-1-yl]-(4-chloro-2-nitrophenyl)methanone NA 500000 NA NA NA NA TTD
BCR 4-[5-Bromo-4-[4-(2,5-dichlorothiophen-3-yl)sulfonylpiperazin-1-yl]pyrimidin-2-yl]morpholine NA 500000 NA NA NA NA TTD
BCR 5-Bromo-2-chloro-4-(4-propylsulfonylpiperazin-1-yl)pyrimidine NA 500000 NA NA NA NA TTD
BDKRB2 (R)-3-Amino-N-(4-aminomethyl-benzyl)-2-{2-[(2-cyclohexyl-acetylamino)-methyl]-pyrrol-1-yl}-propionamide NA NA 101000 NA NA NA BindingDB
BHMT 5-(3-Amino-3-phosphonopropyl)sulfanylpentanoic acid NA 219000 NA NA NA NA BindingDB
BIRC2 2-[(3R)-3-methylpiperazin-1-yl]-1-pyrrolidin-1-ylethanone NA 410000 NA NA NA NA ChEMBL|TTD
BIRC5 N-(4-methylpyridin-2-yl)piperidine-4-carboxamide NA NA 130000 NA NA NA BindingDB
BIRC7 N-{(1s)-1-Cyclohexyl-2-[(2s)-2-(4-Naphthalen-1-Yl-1,3-Thiazol-2-Yl)pyrrolidin-1-Yl]-2-Oxoethyl}-N~2~-Methyl-L-Alaninamide 110000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-1-cyclohexyl-2-oxo-2-((S)-2-(7-phenylthiazolo[5,4-d]pyrimidin-2-yl)pyrrolidin-1-yl)ethyl)-2-(methylamino)propanamide 130000 NA NA NA NA NA BindingDB|TTD
BIRC7 (2S)-N-((1S)-2-((2S)-2-(5-ethynyl-4-(naphthalen-1-yl)thiazol-2-yl)pyrrolidin-1-yl)-2-oxo-1-(tetrahydro-2H-pyran-4-yl)ethyl)-2-(methylamino)propanamide 160000 NA NA NA NA NA BindingDB|TTD
BIRC7 (2S)-2-(methylamino)-N-((1S)-2-((2S)-2-(4-(naphthalen-1-yl)-5-(prop-1-ynyl)thiazol-2-yl)pyrrolidin-1-yl)-2-oxo-1-(tetrahydro-2H-pyran-4-yl)ethyl)propanamide 160000 NA NA NA NA NA BindingDB|TTD
BIRC7 (2S)-N-((1S)-2-((2S)-2-(5-(3-methoxyprop-1-ynyl)-4-(naphthalen-1-yl)thiazol-2-yl)pyrrolidin-1-yl)-2-oxo-1-(tetrahydro-2H-pyran-4-yl)ethyl)-2-(methylamino)propanamide 140000 NA NA NA NA NA BindingDB|TTD
BIRC7 (2S)-N-((1S)-2-((2S)-2-(5-(3-hydroxyprop-1-ynyl)-4-(naphthalen-1-yl)thiazol-2-yl)pyrrolidin-1-yl)-2-oxo-1-(tetrahydro-2H-pyran-4-yl)ethyl)-2-(methylamino)propanamide 140000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-methylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-2-oxoethyl)-2-(methylamino)propanamide 2700000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-isopropylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-2-oxoethyl)-2-(methylamino)propanamide 2800000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-2-((S)-2-(4-benzylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-1-cyclohexyl-2-oxoethyl)-2-(methylamino)propanamide 710000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-1-cyclohexyl-2-oxo-2-((S)-2-(4-(pyridin-3-yl)benzo[d]thiazol-2-yl)pyrrolidin-1-yl)ethyl)-2-(methylamino)propanamide 200000 NA NA NA NA NA BindingDB|TTD
BIRC7 (S)-N-((S)-1-cyclohexyl-2-oxo-2-((S)-2-(4-(pyridin-4-yl)benzo[d]thiazol-2-yl)pyrrolidin-1-yl)ethyl)-2-(methylamino)propanamide 460000 NA NA NA NA NA BindingDB|TTD