| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BLM |
Gabapentin |
NA |
NA |
NA |
NA |
1584890 |
NA |
PubChem |
| BLM |
Ethylmaleimide |
NA |
NA |
NA |
NA |
177828 |
NA |
PubChem |
| BLM |
Propofol |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |
| BLM |
Scopolamine-d3 Hydrobromide |
NA |
NA |
NA |
NA |
6309570 |
NA |
PubChem |
| BLM |
Androstenedione |
NA |
NA |
NA |
NA |
251189 |
NA |
PubChem |
| BLM |
Bupropion Hydrochloride |
NA |
NA |
NA |
NA |
316228 |
NA |
PubChem |
| BLM |
Triflupromazine Hydrochloride |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| BLM |
Orphenadrine Hydrochloride |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |
| BMP1 |
2-[butan-2-yl(4-methoxybenzene)sulfonamido]-N-hydroxyacetamide |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
(S)-2-Acetylamino-5-guanidino-pentanoic acid ((S)-1-hydroxycarbamoyl-ethyl)-amide |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| BMP1 |
(S)-2-Acetylamino-N-hydroxycarbamoylmethyl-3-(4-hydroxy-phenyl)-propionamide |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
2-(N-(2-(hydroxyamino)-2-oxoethyl)-4-methoxyphenylsulfonamido)acetic acid |
NA |
345000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
(4S)-4-[[(2S)-3-carboxy-2-(carboxymethylamino)propanoyl]amino]-5-(methylamino)-5-oxopentanoic acid |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
N-hydroxy-3-[(4-methoxyphenyl)sulfonylamino]propanamide |
NA |
166000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
2-[benzhydryl-(4-methoxyphenyl)sulfonylamino]-N-hydroxyacetamide |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP1 |
Butyl 2-[[2-(hydroxyamino)-2-oxoethyl]-(4-methoxyphenyl)sulfonylamino]acetate |
NA |
167000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BMP4 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4R,5R,6S)-5-acetamido-4-hydroxy-6-pentoxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4,5-dihydroxyoxan-3-yl]oxy-4-hydroxy-5-(sulfonatoamino)-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| BMP4 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-5-acetamido-4-hydroxy-6-pentoxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| BMP4 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-6-(5-aminopentoxy)-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| BMPR1A |
1Kks7U3X86 |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |