| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BMPR1B |
1Kks7U3X86 |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| BMX |
Tak-020 |
NA |
79432800 |
NA |
NA |
NA |
NA |
PubChem |
| BMX |
US9801872, Example 5 |
NA |
79432823 |
NA |
NA |
NA |
NA |
BindingDB |
| BMX |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| BMX |
2-cyano-N-(2,5-dibromophenyl)-3-oxobutanamide |
NA |
281000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
2-Phenyl-octahydropyrrolo(3,4-c)pyrrole |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
6-{4-[3-(dimethylamino)propoxy]phenyl}-2-(methylsulfonyl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-4-amine |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| BPTF |
[1-(3-Fluorophenyl)-3-pyrrolidinyl]methanamine |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
1-(1-Adamantylacetyl)pyrrolidine |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
6-(piperazin-1-yl)-N-(p-tolyl)pyridazin-3-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
6-acetyl-2-amino-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carbonitrile |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
1-[2-(5-Methyl-2-pyridin-3-ylpyrazol-3-yl)oxyphenyl]-3-[4-(trifluoromethoxy)phenyl]urea |
NA |
NA |
6800000 |
NA |
NA |
NA |
BindingDB |
| BPTF |
1-(4-(6-(p-Tolylamino)pyridazin-3-yl)piperazin-1-yl)ethanone |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
3-Chloro-6-(1-piperazinyl)pyridazine |
NA |
750000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
Ipidacrine |
NA |
590000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
4-(Aminomethyl)-1-(3,4-difluorophenyl)pyrrolidin-2-one |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| BPTF |
2-Amino-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carbonitrile |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRAF |
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(2-methoxyphenyl)-N-phenyl-3,4-dihydropyrazole-2-carbothioamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRAF |
5-(4-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-phenyl-3,4-dihydropyrazole-2-carbothioamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRAF |
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-methylphenyl)-N-phenyl-3,4-dihydropyrazole-2-carbothioamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |