| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BRD4 |
N-(4-chloro-3-pyrrolidin-1-ylsulfonylphenyl)acetamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
N-[[1-(1,1-dioxothiolan-3-yl)-3,5-dimethylpyrazol-4-yl]methyl]-N-methyl-3,3-diphenylpropanamide |
NA |
160030 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
Acetaminophen |
NA |
NA |
250000 |
NA |
NA |
NA |
ChEMBL|PubChem |
| BRD4 |
1H-1,5-Benzodiazepin-2-one, 2,3,4,5-tetrahydro-4-methyl- |
NA |
220000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BRD4 |
4-(Hydroxymethyl)-1-methyl-2-pyrrolidinone |
NA |
4110000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BRD4 |
2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
2-Methyl-5-(Methylamino)-6-Phenylpyridazin-3(2h)-One |
160000 |
NA |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| BRD4 |
1-(2-Methyl-3,4-dihydroquinolin-1(2H)-yl)ethan-1-one |
NA |
125892.54 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
3-Phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-amine |
NA |
NA |
109000 |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
3-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
3,4-Dihydro-3-methyl-2(1H)-quinazolinone |
NA |
NA |
102000 |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
4-chloro-2-(7H-purin-6-ylamino)phenol |
NA |
491000 |
NA |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
2-(3,5-Difluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
Ethyl 3-methyl-1,2,3,4-tetrahydro-3-quinolinecarboxylate |
NA |
NA |
610000 |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
Methyl 4-((3-phenylureido)methyl)piperidine-1-carboxylate |
NA |
NA |
270000 |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
(R)-(-)-JQ1 Enantiomer |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
2-(3-methyl-2,5-dioxoimidazolidin-1-yl)-N-(4-methyl-3-piperidin-1-ylsulfonylphenyl)acetamide |
NA |
501187.23 |
NA |
NA |
NA |
NA |
TTD |
| BRD4 |
(4S)-1-methyl-4-phenylpyrrolidin-2-one |
NA |
1430000 |
NA |
NA |
NA |
NA |
ChEMBL |
| BRD4 |
Dimethyl Sulfoxide |
NA |
280000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| BRD4 |
(2S)-2-(hydroxymethyl)-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |