| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BRD9 |
N-[1,4-Dimethyl-7-(morpholin-4-YL)-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-6-YL]-4-(2-methylpropyl)benzene-1-sulfonamide |
NA |
204000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
5-ethyl-5-methyl-5,6-dihydrobenzo[h]quinazolin-4(3H)-one |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
[5-[2-(3,5-Dimethylanilino)pyrimidin-4-yl]-1-piperidin-4-yltriazol-4-yl]methanol |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BRDT |
Methyl 7-thiophen-2-yl-1,4-thiazepane-4-carboxylate |
NA |
NA |
270000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| BRDT |
5-(furan-2-yl)-2-hydroxy-1-(tetrahydrofuran-2-ylmethyl)pyrido[2,3-d]pyrimidin-4(1H)-one |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
8-Chloro-6-(4-chlorophenyl)-1-methyl-3,4-dihydro-1,5-benzodiazocin-2-one |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
2-(3,5-Difluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
1-(4-Chloro-2-phenoxyphenyl)-3-(3,4-dichlorophenyl)urea |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRDT |
Mrs2500 |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRDT |
1-[2-(5-Methyl-2-pyridin-3-ylpyrazol-3-yl)oxyphenyl]-3-[4-(trifluoromethoxy)phenyl]urea |
NA |
NA |
1500000 |
NA |
NA |
NA |
BindingDB |
| BRDT |
1-[2-[2-(2-Ethylphenyl)-5-methylpyrazol-3-yl]oxyphenyl]-3-(4-propan-2-yloxyphenyl)urea |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRDT |
5-{2-[3-(4-tert-butyl-phenyl)-ureido]-phenoxy}-1-phenyl-1H-pyrazole-3-carboxylic acid methyl ester |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRDT |
1-[2-(2-Phenyl-2H-pyrazol-3-yloxy)-phenyl]-3-(4-trifluoromethoxy-phenyl)-urea |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| BRDT |
1,3-Diethyl-2-oxo-2,3-dihydro-1H-benzoimidazole-5-carbaldehyde |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| BRDT |
(E)-N'-methoxy-N-[7-(pyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]methanimidamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| BRPF1 |
3-ethyl-N-[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]pyridine-4-carboxamide |
NA |
515000 |
NA |
NA |
NA |
NA |
TTD |
| BRPF1 |
7-oxo-N-[4-(piperidin-1-ylmethyl)-1,3-thiazol-2-yl]azepane-2-carboxamide |
NA |
293000 |
NA |
NA |
NA |
NA |
TTD |
| BRPF1 |
N-[4-(2-fluoro-5-methoxyphenyl)-1,3-thiazol-2-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRPF1 |
6-{[2-(4-Chlorophenyl)pyrrolidin-1-YL]sulfonyl}-1,4-dimethyl-1,2,3,4-tetrahydroquinoxaline-2,3-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BRPF1 |
6-[3-(2-Ethyl-6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)-3-oxopropyl]sulfonyl-1,4-dimethylquinoxaline-2,3-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |