Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| C1S | 4-Nitrobenzamidine | 92500000|100000000 | NA | NA | NA | NA|NA | NA|NA | BindingDB|TTD |
| C1S | 3-(Dimethylamino)benzenecarboximidamide;2,4,6-trinitrophenol | 199526.23 | NA | NA | NA | NA | NA | TTD |
| C1S | 3-(Phenylmethyl)benzenecarboximidamide | 630000|630957.34 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | 3-Nitrobenzamidinium hydrochloride | 501187.23 | NA | NA | NA | NA | NA | TTD |
| C1S | Phenylguanidine | 548000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | m-Aminobenzamidine hydrochloride | 316000|251188.64 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | Amido Phenyl Pyruvic Acid | 158000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | Aminoguanidine | 18100000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 2-Guanidinoacetate | 4370000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 4-Methoxybenzenecarboximidamide | 100000000 | NA | NA | NA | NA | NA | TTD |
| C1S | Benzamidine | 398000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 3-Amidinophenylpyruvic acid | 251000|100000000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | 3,5-Dimethylbenzenecarboximidamide | 630000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 3-Phenylbenzenecarboximidamide | 7940000|251188.64 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | 3-(Aminoiminomethyl)benzoic acid | 1990000|6309573.44 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | Neopentylguanidine | 13400000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 3-(Hydroxymethyl)benzene-1-carboximidamide | 1580000|10000000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| C1S | [Amino(phenyl)methylidene]azanium | 603000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 3-Bromo-benzamidine | 630000 | NA | NA | NA | NA | NA | BindingDB |
| C1S | 4-Ethoxy-benzamidine | 100000000 | NA | NA | NA | NA | NA | TTD |