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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
C1S 3-Methoxy-benzamidine 160000|158489.32 NA NA NA NA NA BindingDB|TTD
C1S 3,4-Dimethylbenzene-1-carboximidamide 6300000|9990000|125892.54 NA NA NA NA NA BindingDB|TTD
C1S N-z-L-Tyr 370000 NA NA NA NA NA BindingDB
C1S 2-Methyl-benzamidine 1600000|1584893.19 NA NA NA NA NA BindingDB|TTD
C1S 2-[(2-Chloroacetyl)amino]-3-(4-hydroxyphenyl)propanoate 1120000 NA NA NA NA NA BindingDB
C1S [Amino-(3-nitrophenyl)methylidene]azanium;hydrochloride 9990000 NA NA NA NA NA BindingDB
C1S 3-N'-naphthalen-1-ylbenzene-1,3-dicarboximidamide 100000000 NA NA NA NA NA TTD
C1S 2-(3,4-Dihydroquinoxalin-2-yl)guanidine 2970000 NA NA NA NA NA BindingDB
C3 Ac-I[CVVdQDWGHHRC]-NH2 NA 1000000 NA NA NA NA TTD
C3 Ac-Ile-Cys(1)-Val-D-Val-Gln-D-Asp-D-Trp-Gly-His-D-His-Arg-Cys(1)-NH2 NA 1000000 NA NA NA NA TTD
C3AR1 H-Phe-Lys-Pro-Leu-Ala-Ala-D-Ala-Arg-OH NA NA NA 130617 NA NA BindingDB
C3AR1 H-Phe-Leu-Ala-Leu-Ala-Arg-OH NA NA NA 101000 NA NA BindingDB
C5AR1 Tyr-Ser-Phe-Lys-Asp-Cys-Pro-Leu-Cys-Arg NA NA NA 224000 NA NA TTD
C5AR1 Tyr-Ser-Phe-Lys-Asp-Met-Pro-Ala-Gly-Arg NA NA NA 215000 NA NA TTD
C5AR1 Tyr-Ser-Phe-Lys-Asp-Met-Gln-Leu-Pro-Arg NA NA NA 500000 NA NA TTD
C5AR1 (S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-propionylamino)-hexanoyl]-pyrrolidine-2-carbonyl}-amino)-4-methyl-pentanoylamino]-3-(1H-indol-3-yl)-propionylamino]-5-guanidino-pentanoic acid NA 144000 NA NA NA NA TTD
C5AR1 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-cyclohexyl-propionylamino]-3-cyclohexyl-propionylamino}-pentanoylamino)-propionylamino]-5-guanidino-pentanoic acid 600000 NA NA NA NA NA TTD
C5AR1 Acetylhistidyl-lysyl-aspartyl-methionyl-glutaminyl-leucyl-glycyl-arginine 150000 NA NA NA NA NA TTD
C5AR1 Ac-His-Lys-Asp-Nle-Nle-Nle-Gly-Arg-OH 210000 NA NA NA NA NA TTD
C5AR1 2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-3-phenyl-propionylamino]-3-phenyl-propionylamino}-3-phenyl-propionylamino)-propionylamino]-5-guanidino-pentanoic acid 750000 NA NA NA NA NA TTD