| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CA1 |
2-Trifluoromethanesulfonylamino-benzenesulfonamide |
175000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
ethyl 6-(hydroxymethyl)-2-oxo-2H-chromene-3-carboxylate |
213000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
Phosphate Ion |
780000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
4-[2-(2,6-Diphenylpyridin-1-ium-1-yl)ethyl]benzenesulfonamide;perchlorate |
265000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
2,6-Diphenyl-1-[2-(4-sulfamoyl-phenyl)-ethyl]-pyridinium; perchlorate |
265000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
3-Trifluoromethanesulfonylamino-benzenesulfonamide |
188400 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
3-Chloro-4-trifluoromethanesulfonylamino-benzenesulfonamide |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
4-[(2-Tert-butyl-4,6-diphenylpyridin-1-ium-1-yl)methyl]benzenesulfonamide;perchlorate |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
2-tert-Butyl-4,6-diphenyl-1-(4-sulfamoyl-benzyl)-pyridinium; perchlorate |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
4-(2,4-Diphenyl-6-propan-2-ylpyridin-1-ium-1-yl)benzenesulfonamide;perchlorate |
125000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
2-Isopropyl-4,6-diphenyl-1-(4-sulfamoyl-phenyl)-pyridinium; perchlorate |
125000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
3-Iodo-4-trifluoromethanesulfonylamino-benzenesulfonamide |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
4-[(2,6-Diphenylpyridin-1-ium-1-yl)methyl]benzenesulfonamide;perchlorate |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
4-[(2,6-Diphenylpyridin-1-ium-1-yl)methyl]benzenesulfonamide |
280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
4-[2-(2,4,6-Triphenylpyridin-1-ium-1-yl)ethyl]benzenesulfonamide;perchlorate |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
4-[2-(2,4,6-Triphenylpyridin-1-ium-1-yl)ethyl]benzenesulfonamide |
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Trifluoro-methanesulfonic acid 4-sulfamoyl-benzyl ester |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
4-(2,4,6-Triphenylpyridin-1-ium-1-yl)benzenesulfonamide;perchlorate |
290000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
3-Bromo-4-trifluoromethanesulfonylamino-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
Syringic acid |
919000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |